Protein kinase cAMP-activated catalytic subunit alpha
Kinase structure
Kinase:PRKACA (PKACa)
Family:PKA
Group:AGC
Species:HUMAN
IUPHAR/BPS ID:1476
PDB:5J5X
sc-PDB:
KIDFamMap:Search
Release date:2016-07-20
PubMed: 27389935
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 5J5X
5J5XAlternative model: AChain: A
5J5XAlternative model: CChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):56.8° (17.5Å)
G-rich loop rotation:49.2°
Quality Score:8
Resolution:2.6 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I10
Ligand
No
Protein
No

Allosteric Ligand
Allosteric ligand:6J9
2D structure of the allostericligand
Pocket alignment
Uniprot sequence:KTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVPGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA
Sequence structure:KTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVPGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA