Mitogen-activated protein kinase kinase kinase 5
Kinase structure
Kinase:MAP3K5
Family:STE11
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2080
PDB:5VIO
sc-PDB:
KIDFamMap:Search
Release date:2018-01-17
PubMed: 29348070
Chain:C
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The orthosteric binding pocket


More entries for 5VIO
5VIOChain: A
5VIOChain: B
5VIOChain: D


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):50.1° (14.7Å)
G-rich loop rotation:75.4°
Quality Score:8
Resolution:2.84 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I7
I11
Ligand
No
No
Protein
No
No

Pocket alignment
Uniprot sequence:VVLGKGTYGIVYAIAIKEIPLHEEIALHKHLKKNIVQYLGSKIFMEQVPGGSLSALLRSYLHDNQIVHRDIKGDNVLIISDFGTS
Sequence structure:VVLGKGTYGIVYAIAIKEIPLHEEIALHKHLKKNIVQYLGSKIFMEQVPGGSLSALLRSYLHDNQIVHRDIKGDNVLIISDFGTS