PDB-code
Browse kinase entries (page 115 of 282)
First 111 112 113 PreviousLast119 118 117 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | EPHA3 (EphA3) | Eph | TK | 4g2f | A | A | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4g2f | A | B | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk3 | A | A | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk3 | A | B | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk4 | A | A | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4gk4 | A | B | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4p4c | A | 2-amino-1-(3-methoxyphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() | |
![]() | EPHA3 (EphA3) | Eph | TK | 4p5q | A | A | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4p5q | A | B | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4p5z | A | 2-amino-1-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | Show | ![]() | |
![]() | EPHA3 (EphA3) | Eph | TK | 4twn | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4twn | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4two | A | A | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 4two | A | B | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 6in0 | A | A | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | Show | ![]() |
![]() | EPHA3 (EphA3) | Eph | TK | 6in0 | A | B | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | Show | ![]() |
![]() | Epha4 (EphA4) | Eph | TK | 2hel | A | - | Mouse | Show | ![]() | |
![]() | Epha4 (EphA4) | Eph | TK | 2xyu | A | 5-(5-fluoro-2-methylphenyl)-6,7,8,9-tetrahydro-3h-pyrazolo[3,4-c]isoquinolin-1-amine | Mouse | Show | ![]() | |
![]() | Epha4 (EphA4) | Eph | TK | 2y6m | A | A | - | Mouse | Show | ![]() |
![]() | Epha4 (EphA4) | Eph | TK | 2y6m | A | B | - | Mouse | Show | ![]() |
![]() | Epha4 (EphA4) | Eph | TK | 2y6o | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | Show | ![]() |
![]() | Epha4 (EphA4) | Eph | TK | 2y6o | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | Show | ![]() |
![]() | EPHA5 (EphA5) | Eph | TK | 2r2p | A | A | - | Human | Show | ![]() |
![]() | EPHA5 (EphA5) | Eph | TK | 2r2p | A | B | - | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 2rei | A | A | - | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 2rei | A | B | - | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 3dko | A | A | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 3dko | A | B | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 7eec | A | A | - | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 7eec | A | B | - | Human | Show | ![]() |
![]() | EPHA7 (EphA7) | Eph | TK | 7eed | A | - | Human | Show | ![]() | |
![]() | EPHA7 (EphA7) | Eph | TK | 7eef | A | - | Human | Show | ![]() | |
![]() | EPHA8 (EphA8) | Eph | TK | 3kul | A | A | - | Human | Show | ![]() |
![]() | EPHA8 (EphA8) | Eph | TK | 3kul | A | B | - | Human | Show | ![]() |
![]() | EPHA8 (EphA8) | Eph | TK | 3kul | B | A | - | Human | Show | ![]() |
![]() | EPHA8 (EphA8) | Eph | TK | 3kul | B | B | - | Human | Show | ![]() |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | A | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | B | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | C | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | D | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | E | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | F | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | G | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | H | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 3zfx | I | - | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 5mja | A | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 5mja | B | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | Show | ![]() | |
![]() | EPHB1 (EphB1) | Eph | TK | 5mjb | A | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | Show | ![]() |


