PDB-code
Browse kinase entries (page 117 of 282)
First 113 114 115 PreviousLast121 120 119 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | EPHB4 (EphB4) | Eph | TK | 6fni | A | B | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | Show |  |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | A | - | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | B | - | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | A | A | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | A | B | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | B | A | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | B | B | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | A | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | Show | | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | B | - | Human | Show | | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | C | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | Show | | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | D | - | Human | Show | | |
| ERBB2 (ErbB2) | EGFR | TK | 7jxh | A | A | (2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamide | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 7jxh | A | B | (2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamide | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 7pcd | A | A | 1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-one | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 7pcd | A | B | 1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-one | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 8u8x | A | A | 1-{(1r,3r,5s)-3-[(3m)-4-methyl-3-{3-methyl-4-[(1-methyl-1h-benzimidazol-5-yl)oxy]phenyl}-1h-pyrazolo[3,4-d]pyrimidin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl}propan-1-one | Human | Show | |
| ERBB2 (ErbB2) | EGFR | TK | 8u8x | A | B | 1-{(1r,3r,5s)-3-[(3m)-4-methyl-3-{3-methyl-4-[(1-methyl-1h-benzimidazol-5-yl)oxy]phenyl}-1h-pyrazolo[3,4-d]pyrimidin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl}propan-1-one | Human | Show | |
| ERBB3 (ErbB3) | EGFR | TK | 3kex | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 3kex | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 3lmg | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 3lmg | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4riw | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4riw | C | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4rix | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4rix | C | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4riy | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 4riy | C | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 6op9 | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | |
| ERBB3 (ErbB3) | EGFR | TK | 6op9 | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | Show | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn5 | A | - | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn6 | A | - | Human | Show | | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn8 | A | - | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | Show | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | Show | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | Show | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | Show | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | D | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbw | A | - | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbw | B | - | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 3bce | A | - | Human | Show | | |
| ERBB4 (ErbB4) | EGFR | TK | 3bce | B | - | Human | Show | |
