Browse kinase entries (page 125 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
FGFR2FGFRTK4j99CAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK4j99CBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK4j99CCphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK4j99DAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK4j99DBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK4j99DCphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5eg3Aphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5uglAAphosphoaminophosphonic acid-adenylate esterHumanShow
FGFR2FGFRTK5uglABphosphoaminophosphonic acid-adenylate esterHumanShow
FGFR2FGFRTK5uglBAphosphoaminophosphonic acid-adenylate esterHumanShow
FGFR2FGFRTK5uglBBphosphoaminophosphonic acid-adenylate esterHumanShow
FGFR2FGFRTK5ugxAAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5ugxABphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5ugxBAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5ugxBBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5uhnAAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5uhnABphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5uhnBAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5uhnBBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5ui0AA-HumanShow
FGFR2FGFRTK5ui0AB-HumanShow
FGFR2FGFRTK5ui0BAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK5ui0BBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK6agxAAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxABethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxBAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxBBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxCAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxCBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxDAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6agxDBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHumanShow
FGFR2FGFRTK6lvkAn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHumanShow
FGFR2FGFRTK6lvkBn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHumanShow
FGFR2FGFRTK6lvlAn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHumanShow
FGFR2FGFRTK6lvlBn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHumanShow
FGFR2FGFRTK6v6qAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK6v6qBphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK6v6qCphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK6v6qDphosphomethylphosphonic acid adenylate esterHumanShow
FGFR2FGFRTK7kiaAA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHumanShow
FGFR2FGFRTK7kiaAB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHumanShow
FGFR2FGFRTK7kiaBA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHumanShow
FGFR2FGFRTK7kiaBB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHumanShow
FGFR2FGFRTK7kieAAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHumanShow
FGFR2FGFRTK7kieABn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHumanShow
FGFR2FGFRTK7kieBAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHumanShow
FGFR2FGFRTK7kieBBn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHumanShow
FGFR2FGFRTK7ozyAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHumanShow
FGFR2FGFRTK7ozyAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHumanShow
FGFR2FGFRTK8e1xA(5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamideHumanShow
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