PDB-code
Browse kinase entries (page 125 of 282)
First 121 122 123 PreviousLast129 128 127 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | FGFR2 | FGFR | TK | 4j99 | C | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 4j99 | C | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 4j99 | C | C | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 4j99 | D | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 4j99 | D | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 4j99 | D | C | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5eg3 | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 5ugl | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugl | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugl | B | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugl | B | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugx | A | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugx | A | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugx | B | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ugx | B | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5uhn | A | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5uhn | A | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5uhn | B | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5uhn | B | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ui0 | A | A | - | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ui0 | A | B | - | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ui0 | B | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 5ui0 | B | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | A | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | A | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | B | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | B | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | C | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | C | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | D | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6agx | D | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 6lvk | A | n-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6lvk | B | n-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6lvl | A | n-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6lvl | B | n-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6v6q | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6v6q | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6v6q | C | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 6v6q | D | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR2 | FGFR | TK | 7kia | A | A | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kia | A | B | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kia | B | A | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kia | B | B | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kie | A | A | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kie | A | B | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kie | B | A | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7kie | B | B | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7ozy | A | A | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 7ozy | A | B | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | Show | ![]() |
![]() | FGFR2 | FGFR | TK | 8e1x | A | (5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamide | Human | Show | ![]() |


