PDB-code
Browse kinase entries (page 135 of 282)
First 131 132 133 PreviousLast139 138 137 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | HASPIN (Haspin) | Haspin | Other | 6z5d | A | B | 11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | Show |  |
| HASPIN (Haspin) | Haspin | Other | 6z5e | A | A | 11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 6z5e | A | B | 11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 7avq | A | A | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 7avq | A | B | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 7ops | A | 2-methylsulfanyl-10-nitro-pyrido[3,4-g]quinazoline | Human | Show | | |
| HASPIN (Haspin) | Haspin | Other | 7sqm | A | A | 1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amine | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 7sqm | A | B | 1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amine | Human | Show | |
| HASPIN (Haspin) | Haspin | Other | 8rdk | A | 3-pyridin-4-yl-1~{h}-pyrrolo[3,2-g]isoquinoline | Human | Show | | |
| HCK | Src | TK | 1ad5 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| HCK | Src | TK | 1ad5 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| HCK | Src | TK | 1qcf | A | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | Show | | |
| HCK | Src | TK | 2c0i | A | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0i | A | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0i | B | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0i | B | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0o | A | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0o | A | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0o | B | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0o | B | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0t | A | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0t | A | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0t | B | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2c0t | B | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | Show | |
| HCK | Src | TK | 2hck | A | 3,5,7,3',4'-pentahydroxyflavone | Human | Show | | |
| HCK | Src | TK | 2hck | B | 3,5,7,3',4'-pentahydroxyflavone | Human | Show | | |
| HCK | Src | TK | 2hk5 | A | 3-{[2-(1h-benzimidazol-1-yl)-6-{[2-(diethylamino)ethyl]amino}pyrimidin-4-yl]amino}-4-methylphenol | Human | Show | | |
| HCK | Src | TK | 3vry | A | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | Show | | |
| HCK | Src | TK | 3vry | B | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | Show | | |
| HCK | Src | TK | 3vrz | A | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | Show | | |
| HCK | Src | TK | 3vrz | B | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | Show | | |
| HCK | Src | TK | 3vs0 | A | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | Show | | |
| HCK | Src | TK | 3vs0 | B | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | Show | | |
| HCK | Src | TK | 3vs1 | A | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | Show | | |
| HCK | Src | TK | 3vs1 | B | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | Show | | |
| HCK | Src | TK | 3vs2 | A | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs2 | B | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs3 | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs3 | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs4 | A | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs4 | B | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs5 | A | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs5 | B | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs6 | A | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | Show | | |
| HCK | Src | TK | 3vs6 | B | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | Show | | |
| HCK | Src | TK | 3vs7 | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 3vs7 | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | | |
| HCK | Src | TK | 4lud | A | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | Show | | |
| HCK | Src | TK | 4lud | B | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | Show | | |
| HCK | Src | TK | 4lue | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | |
