PDB-code
Browse kinase entries (page 160 of 282)
First 156 157 158 PreviousLast164 163 162 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | KIT | PDGFR | TK | 6xva | A | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | Show |  | |
| KIT | PDGFR | TK | 6xva | B | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | Show | | |
| KIT | PDGFR | TK | 6xvb | A | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | Show | | |
| KIT | PDGFR | TK | 6xvb | B | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | Show | | |
| KIT | PDGFR | TK | 7khg | A | A | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | Show | |
| KIT | PDGFR | TK | 7khg | A | B | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | Show | |
| KIT | PDGFR | TK | 7khj | A | 2-phenyl-5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | Show | | |
| KIT | PDGFR | TK | 7khk | A | 4,5-dimethyl-n-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazole-3-carboxamide | Human | Show | | |
| KIT | PDGFR | TK | 7zw8 | A | A | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | Show | |
| KIT | PDGFR | TK | 7zw8 | A | B | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | Show | |
| KIT | PDGFR | TK | 7zy6 | A | 5-imidazo[1,2-a]pyridin-3-yl-~{n}-[(1~{r})-1-(6-pyrrolidin-1-ylpyridin-3-yl)ethyl]pyridin-3-amine | Human | Show | | |
| KIT | PDGFR | TK | 8dfm | A | - | Human | Show | | |
| KIT | PDGFR | TK | 8dfp | A | - | Human | Show | | |
| KIT | PDGFR | TK | 8dfq | A | - | Human | Show | | |
| KIT | PDGFR | TK | 8pq9 | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pq9 | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqa | A | A | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | Show | |
| KIT | PDGFR | TK | 8pqa | A | B | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | Show | |
| KIT | PDGFR | TK | 8pqb | A | A | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqb | A | B | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqc | A | A | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqc | A | B | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqd | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | Show | |
| KIT | PDGFR | TK | 8pqd | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | Show | |
| KIT | PDGFR | TK | 8pqe | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | Show | |
| KIT | PDGFR | TK | 8pqe | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | Show | |
| KIT | PDGFR | TK | 8pqf | A | A | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | Show | |
| KIT | PDGFR | TK | 8pqf | A | B | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | Show | |
| KIT | PDGFR | TK | 8pqg | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KIT | PDGFR | TK | 8pqg | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | Show | |
| KSR1 | RAF | TKL | 7juw | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7jux | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7juy | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7juz | A | - | Human | Show | | |
| KSR1 | RAF | TKL | 7juz | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7jv0 | A | - | Human | Show | | |
| KSR1 | RAF | TKL | 7jv0 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7jv1 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR1 | RAF | TKL | 7jv1 | D | - | Human | Show | | |
| KSR2 | RAF | TKL | 2y4i | B | adenosine-5'-triphosphate | Human | Show | | |
| KSR2 | RAF | TKL | 5kkr | B | 6,7-dimethoxy-~{n}-(2-methyl-4-phenoxy-phenyl)quinazolin-4-amine | Human | Show | | |
| KSR2 | RAF | TKL | 7juq | B | adenosine-5'-diphosphate | Human | Show | | |
| KSR2 | RAF | TKL | 7jur | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR2 | RAF | TKL | 7jus | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR2 | RAF | TKL | 7jut | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR2 | RAF | TKL | 7juu | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| KSR2 | RAF | TKL | 7juv | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| LCK | Src | TK | 1qpc | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| LCK | Src | TK | 1qpd | A | staurosporine | Human | Show | | |
| LCK | Src | TK | 1qpe | A | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | Show | |
