PDB-code
Browse kinase entries (page 167 of 282)
First 163 164 165 PreviousLast171 170 169 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAP2K7 | STE7 | STE | 7ovj | A | A | 1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show |  |
| MAP2K7 | STE7 | STE | 7ovj | A | B | 1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovk | A | 1-[(3~{r})-3-[4-azanyl-3-[1-(5-bromanyl-2-oxidanyl-phenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | Show | | |
| MAP2K7 | STE7 | STE | 7ovl | A | A | 3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovl | A | B | 3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovm | A | A | ~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamide | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovm | A | B | ~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamide | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovn | A | A | 3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | Show | |
| MAP2K7 | STE7 | STE | 7ovn | A | B | 3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | A | - | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | B | - | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | A | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | B | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | A | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | B | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | A | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | B | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | A | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | B | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | A | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | B | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8deg | A | methyl (1s,4s)-5-{(4p)-4-[5-amino-6-(difluoromethoxy)pyrazin-2-yl]-6-[(1r,4r)-2-azabicyclo[2.1.1]hexan-2-yl]pyridin-2-yl}-2,5-diazabicyclo[2.2.1]heptane-2-carboxylate | Human | Show | | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | A | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | B | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | A | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | B | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | A | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | Show | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | B | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | A | - | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | B | - | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | A | - | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | B | - | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | A | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | B | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | A | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | B | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | |
