PDB-code
Browse kinase entries (page 170 of 282)
First 166 167 168 PreviousLast174 173 172 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAP3K5 | STE11 | STE | 5vil | D | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | Show |  | |
| MAP3K5 | STE11 | STE | 5vio | A | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 5vio | B | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 5vio | C | - | Human | Show | | |
| MAP3K5 | STE11 | STE | 5vio | D | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2m | A | n-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2m | B | n-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2n | A | n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2n | B | n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2o | A | 4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6e2o | B | 4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6oyt | A | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6oyt | B | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6oyt | C | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6oyt | D | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | Show | | |
| MAP3K5 | STE11 | STE | 6oyw | A | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | A | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | B | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | B | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | C | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | C | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | D | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6oyw | D | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | Show | |
| MAP3K5 | STE11 | STE | 6vre | A | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6vre | A | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6vre | B | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6vre | B | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6xih | A | A | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6xih | A | B | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6xih | B | A | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 6xih | B | B | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 7mu7 | A | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 7mu7 | A | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | Show | |
| MAP3K5 | STE11 | STE | 8qgy | A | - | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | A | adenosine | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | B | adenosine | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 2yiy | A | (1e)-1-[5-tert-butyl-2-(3-fluorophenyl)-1h-pyrazol-3-ylidene]-3-(4-pyridin-3-yloxyphenyl)urea | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | A | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | B | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4l3p | A | 2-(1-benzothiophen-7-yl)-4-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[2,3-c]pyridin-7-amine | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | A | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | B | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | A | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | B | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | Show | |
| MAP3K7 (TAK1) | MLK | TKL | 4o91 | A | n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methyl-3-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5e7r | A | 2-chloro-n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}acetamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjd | A | 1-(4-((1h-pyrrolo[2,3-b]pyridin-4-yl)oxy)phenyl)-3-(5-(4-methylpiperazin-1-yl)naphthalen-2-yl)urea | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjf | A | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(3-phenylureido)phenyl)thiazole-4-carboxamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjg | A | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(phenylcarbamoyl)phenyl)thiazole-4-carboxamide | Human | Show | | |
| MAP3K7 (TAK1) | MLK | TKL | 5j7s | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | Show | |
