Browse kinase entries (page 18 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
AURKA (AurA)AurOther4jbqAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHumanShow
AURKA (AurA)AurOther4o0sAadenosineHumanShow
AURKA (AurA)AurOther4o0uAadenosineHumanShow
AURKA (AurA)AurOther4o0wAadenosineHumanShow
AURKA (AurA)AurOther4prjAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHumanShow
AURKA (AurA)AurOther4uynAethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther4uzdAethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther4uzdBethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther4uzhA(4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-oneHumanShow
AURKA (AurA)AurOther4zs0A5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-oneHumanShow
AURKA (AurA)AurOther4ztqA(2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-oneHumanShow
AURKA (AurA)AurOther4ztrA6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acidHumanShow
AURKA (AurA)AurOther4ztsA(2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-oneHumanShow
AURKA (AurA)AurOther5aadA7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther5aaeA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazoleHumanShow
AURKA (AurA)AurOther5aafA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamideHumanShow
AURKA (AurA)AurOther5aagA[3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanoneHumanShow
AURKA (AurA)AurOther5dn3AAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dn3ABadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dnrAAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dnrABadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dosAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dpvAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dpvAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dr2Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dr6AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dr6AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dr9A4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5drdAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dt0AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dt0AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dt3Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dt4Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5ew9AA4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHumanShow
AURKA (AurA)AurOther5ew9AB4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHumanShow
AURKA (AurA)AurOther5g15AAphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther5g15ABphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther5g1xAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5g1xABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8jAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8jABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8kAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8kABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8lAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8lABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5lxmAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5lxmABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5objAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5obrA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5odtAAadenosine-5'-diphosphateHumanShow
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