Browse kinase entries (page 174 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAP4K4 (HGK)STE20STE4zp5B-HumanShow
MAP4K4 (HGK)STE20STE5di1A4-{6-amino-5-[4-(methylsulfonyl)phenyl]pyridin-3-yl}phenolHumanShow
MAP4K4 (HGK)STE20STE5di1B-HumanShow
MAP4K4 (HGK)STE20STE5j95A1-{4-[6-amino-5-(4-chlorophenyl)pyridin-3-yl]phenyl}cyclopentane-1-carboxylic acidHumanShow
MAP4K4 (HGK)STE20STE5j95B-HumanShow
MAP4K4 (HGK)STE20STE5w5qAA(5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideHumanShow
MAP4K4 (HGK)STE20STE5w5qAB(5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideHumanShow
MAP4K4 (HGK)STE20STE5w5qBA-HumanShow
MAP4K4 (HGK)STE20STE5w5qBB-HumanShow
MAPK1 (Erk2)MAPKCMGC1pmeA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHumanShow
MAPK1 (Erk2)MAPKCMGC1tvoA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHumanShow
MAPK1 (Erk2)MAPKCMGC1wzyA1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHumanShow
MAPK1 (Erk2)MAPKCMGC2ojgAn,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC2ojiAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC2ojjA(s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC2y9qAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC2y9qABphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC2y9qACphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC3i5zAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC3i60A4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC3sa0AAnorathyriolHumanShow
MAPK1 (Erk2)MAPKCMGC3sa0ABnorathyriolHumanShow
MAPK1 (Erk2)MAPKCMGC3teiAphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC3w55A(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHumanShow
MAPK1 (Erk2)MAPKCMGC4fmqAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC4fmqABphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK1 (Erk2)MAPKCMGC4fuxAtrans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanolHumanShow
MAPK1 (Erk2)MAPKCMGC4fuyAA{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHumanShow
MAPK1 (Erk2)MAPKCMGC4fuyAB{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHumanShow
MAPK1 (Erk2)MAPKCMGC4fv0AAn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHumanShow
MAPK1 (Erk2)MAPKCMGC4fv0ABn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHumanShow
MAPK1 (Erk2)MAPKCMGC4fv1AAn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv1ABn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv2AA4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv2AB4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv3AAethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHumanShow
MAPK1 (Erk2)MAPKCMGC4fv3ABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHumanShow
MAPK1 (Erk2)MAPKCMGC4fv4AA9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHumanShow
MAPK1 (Erk2)MAPKCMGC4fv4AB9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHumanShow
MAPK1 (Erk2)MAPKCMGC4fv5An-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv6An-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHumanShow
MAPK1 (Erk2)MAPKCMGC4fv7AA4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHumanShow
MAPK1 (Erk2)MAPKCMGC4fv7AB4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHumanShow
MAPK1 (Erk2)MAPKCMGC4fv8AA6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHumanShow
MAPK1 (Erk2)MAPKCMGC4fv8AB6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHumanShow
MAPK1 (Erk2)MAPKCMGC4fv9AA3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHumanShow
MAPK1 (Erk2)MAPKCMGC4fv9AB3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHumanShow
MAPK1 (Erk2)MAPKCMGC4g6nAA3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHumanShow
MAPK1 (Erk2)MAPKCMGC4g6nAB3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHumanShow
MAPK1 (Erk2)MAPKCMGC4g6oA4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHumanShow
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