PDB-code
Browse kinase entries (page 179 of 282)
First 175 176 177 PreviousLast183 182 181 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | B | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | A | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | B | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | A | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | B | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | A | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | B | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | A | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | B | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | A | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | B | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | A | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | B | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | A | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | B | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | A | 1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-one | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8psy | A | - | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | A | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | B | - | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8u8j | A | (4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 8u8k | A | (4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 1jnk | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 1pmn | A | cyclopropyl-{4-[5-(3,4-dichlorophenyl)-2-[(1-methyl)-piperidin]-4-yl-3-propyl-3h-imidazol-4-yl]-pyrimidin-2-yl}amine | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 1pmu | A | 9-(4-hydroxyphenyl)-2,7-phenanthroline | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 1pmv | A | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2b1p | A | 3-{6-[(2-chlorophenyl)amino]-1h-indazol-3-yl}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acid | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2exc | X | n-{2'-[(4-fluorophenyl)amino]-4,4'-bipyridin-2-yl}-4-methoxycyclohexanecarboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2o0u | A | n-{3-cyano-6-[3-(1-piperidinyl)propanoyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl}1-naphthalenecarboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2o2u | A | n-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | A | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | B | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2p33 | A | 4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2r9s | A | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2r9s | B | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | A | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | B | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | A | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | Show | ![]() |


