Browse kinase entries (page 180 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAPK10 (JNK3)MAPKCMGC2zdtAB4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acidHumanShow
MAPK10 (JNK3)MAPKCMGC2zduA4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acidHumanShow
MAPK10 (JNK3)MAPKCMGC3cgfAn-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC3cgoA2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamideHumanShow
MAPK10 (JNK3)MAPKCMGC3da6An-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amineHumanShow
MAPK10 (JNK3)MAPKCMGC3fi2AA3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3fi2AB3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3fi3AA3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3fi3AB3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3fv8AA5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC3fv8AB5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHumanShow
MAPK10 (JNK3)MAPKCMGC3g90X(3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oximeHumanShow
MAPK10 (JNK3)MAPKCMGC3g9lX(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oximeHumanShow
MAPK10 (JNK3)MAPKCMGC3g9nA(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oximeHumanShow
MAPK10 (JNK3)MAPKCMGC3kvxAAn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHumanShow
MAPK10 (JNK3)MAPKCMGC3kvxABn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHumanShow
MAPK10 (JNK3)MAPKCMGC3oxiAmethyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylateHumanShow
MAPK10 (JNK3)MAPKCMGC3oy1A5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHumanShow
MAPK10 (JNK3)MAPKCMGC3ptgAn-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHumanShow
MAPK10 (JNK3)MAPKCMGC3rtpAn-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHumanShow
MAPK10 (JNK3)MAPKCMGC3ttiAtrans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanolHumanShow
MAPK10 (JNK3)MAPKCMGC3ttjAA9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHumanShow
MAPK10 (JNK3)MAPKCMGC3ttjAB9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHumanShow
MAPK10 (JNK3)MAPKCMGC3v6rAA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3v6rAB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3v6rBA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3v6rBB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3v6sAB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC3v6sBB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4h36AA-HumanShow
MAPK10 (JNK3)MAPKCMGC4h36AB-HumanShow
MAPK10 (JNK3)MAPKCMGC4h39AA-HumanShow
MAPK10 (JNK3)MAPKCMGC4h39AB-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bAA-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bAB-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bAC-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bCA-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bCB-HumanShow
MAPK10 (JNK3)MAPKCMGC4h3bCC-HumanShow
MAPK10 (JNK3)MAPKCMGC4kkeAadenosine monophosphateHumanShow
MAPK10 (JNK3)MAPKCMGC4kkgA-HumanShow
MAPK10 (JNK3)MAPKCMGC4kkhAcyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanoneHumanShow
MAPK10 (JNK3)MAPKCMGC4u79An-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamideHumanShow
MAPK10 (JNK3)MAPKCMGC4w4vA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4w4wAn-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4w4xA3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4w4yA3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4whzAA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4whzAB3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHumanShow
MAPK10 (JNK3)MAPKCMGC4x21An-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHumanShow
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