PDB-code
Browse kinase entries (page 180 of 282)
First 176 177 178 PreviousLast184 183 182 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
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![]() | MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | B | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 2zdu | A | 4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acid | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3cgf | A | n-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amine | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3cgo | A | 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3da6 | A | n-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amine | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | A | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | B | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | A | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | B | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | A | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | B | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3g90 | X | (3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oxime | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3g9l | X | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oxime | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3g9n | A | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oxime | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | A | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | B | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3oxi | A | methyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylate | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3oy1 | A | 5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3ptg | A | n-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3rtp | A | n-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3tti | A | trans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanol | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | A | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | B | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6s | A | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 3v6s | B | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | A | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | B | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | A | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | B | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | A | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | B | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | C | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | A | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | B | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | C | - | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4kke | A | adenosine monophosphate | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4kkg | A | - | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4kkh | A | cyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanone | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4u79 | A | n-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4w4v | A | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4w4w | A | n-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4w4x | A | 3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4w4y | A | 3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | Show | ![]() | |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | A | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | B | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | Show | ![]() |
![]() | MAPK10 (JNK3) | MAPK | CMGC | 4x21 | A | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | Show | ![]() |


