PDB-code
Browse kinase entries (page 182 of 282)
First 178 179 180 PreviousLast186 185 184 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK13 (p38d) | MAPK | CMGC | 3coi | A | B | - | Human | Show | ![]() |
![]() | MAPK13 (p38d) | MAPK | CMGC | 4eyj | A | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]urea | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 4eym | A | 2-(morpholin-4-yl)-n-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamide | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 4myg | A | - | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 4myg | B | - | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 4yno | A | - | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 5ekn | A | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]urea | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 5eko | A | 3-(4-methyl-1h-imidazol-1-yl)-n-[4-(pyridin-4-yloxy)phenyl]benzamide | Human | Show | ![]() | |
![]() | MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | A | - | Human | Show | ![]() |
![]() | MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | B | - | Human | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 1lew | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 1lez | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 1yw2 | A | 2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-one | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 1ywr | A | 4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-one | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2ghl | A | 3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2ghm | A | 3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2gtm | A | 8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diium | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2gtn | A | 2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amine | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2oza | B | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 2puu | A | 5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-ium | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p4k | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p5k | A | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p78 | A | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylurea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p79 | A | 1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylurea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p7a | A | 1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylurea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p7b | A | 1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3p7c | A | 1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3py3 | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 3tg1 | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4ka3 | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loo | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loo | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4lop | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 4loq | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |


