PDB-code
Browse kinase entries (page 185 of 282)
First 181 182 183 PreviousLast189 188 187 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | B | 2-phenoxyacetamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | A | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | B | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | A | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | B | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | A | 4-methylbenzamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | B | 4-methylbenzamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | A | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | B | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | A | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | B | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 5uoj | A | - | Mouse | Show | ![]() | |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sod | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sod | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6soi | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6soi | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sot | A | A | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sot | A | B | - | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sou | A | A | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sou | A | B | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sov | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sov | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6spl | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6spl | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | A | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |
![]() | Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | B | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | Show | ![]() |


