PDB-code
Browse kinase entries (page 188 of 282)
First 184 185 186 PreviousLast192 191 190 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK14 (p38a) | MAPK | CMGC | 2okr | D | - | Human | Show |  | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | B | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2qd9 | A | 1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg5 | A | n-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg6 | A | 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2yis | A | 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2yiw | A | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2yix | A | 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | A | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | B | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | A | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | B | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | A | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | B | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv2 | A | 5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv3 | A | 5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3bx5 | A | n-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3c5u | A | 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ctq | A | n-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | A | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | B | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3d83 | A | n-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | A | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | B | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | C | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | D | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3dt1 | A | n-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3e92 | A | n-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | A | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | B | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fc1 | X | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fi4 | A | (2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkl | A | n-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkn | A | 3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fko | A | 3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fl4 | A | 6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fln | C | 6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flq | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fls | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flw | A | 6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fly | A | 6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flz | A | 8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmh | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmj | A | 4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmk | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fml | A | 6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmm | A | 6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | |
