PDB-code
Browse kinase entries (page 194 of 282)
First 190 191 192 PreviousLast198 197 196 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | Show |  |
| MAPK14 (p38a) | MAPK | CMGC | 8a8m | A | phosphomethylphosphonic acid adenosyl ester | Human | Show | | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | Show | | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | Show | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | A | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | B | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | C | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | D | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | A | ~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamine | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | B | - | Human | Show | | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | A | - | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | B | - | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | A | - | Human | Show | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | B | - | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 4b99 | A | 11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | D | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | A | - | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | B | - | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | A | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | B | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | A | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | B | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsl | A | 3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamide | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | A | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | B | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | A | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | B | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | A | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | B | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkm | A | [4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanone | Human | Show | | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | A | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | B | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | Show | |
| MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | A | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | Show | |
