PDB-code
Browse kinase entries (page 200 of 282)
First 196 197 198 PreviousLast204 203 202 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MELK | CAMKL | CAMK | 4d2p | D | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | A | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | A | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | B | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | B | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | C | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | C | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | D | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2t | D | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | A | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | A | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | B | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | B | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | C | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | C | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | D | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2v | D | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | A | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | A | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | B | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | B | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | C | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | C | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | D | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4d2w | D | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ixp | A | - | Human | Show | ![]() | |
![]() | MELK | CAMKL | CAMK | 4ump | A | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | A | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | B | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | B | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | C | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | C | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | D | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4ump | D | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4umq | A | A | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4umq | A | B | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 4umr | A | 4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide | Human | Show | ![]() | |
![]() | MELK | CAMKL | CAMK | 4umt | A | 1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediium | Human | Show | ![]() | |
![]() | MELK | CAMKL | CAMK | 4umu | A | (2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminium | Human | Show | ![]() | |
![]() | MELK | CAMKL | CAMK | 5ih8 | A | n-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamide | Human | Show | ![]() | |
![]() | MELK | CAMKL | CAMK | 5ih9 | A | A | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5ih9 | A | B | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5iha | A | A | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5iha | A | B | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5ihc | A | A | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5ihc | A | B | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5k00 | A | A | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5k00 | A | B | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5m5a | A | A | k-252a | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 5m5a | A | B | k-252a | Human | Show | ![]() |


