PDB-code
Browse kinase entries (page 230 of 282)
First 226 227 228 PreviousLast234 233 232 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PIM1 | PIM | CAMK | 4as0 | A | B | phtalimide-ruthenium complex | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4bzn | A | n-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4bzo | A | n-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4dtk | A | A | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4dtk | A | B | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4enx | A | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4eny | A | A | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4eny | A | B | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4gw8 | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4gw8 | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4i41 | A | 1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedione | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4iaa | A | 10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4jx3 | A | - | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4jx7 | A | 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4k0y | A | A | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4k0y | A | B | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4k18 | A | 5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4k1b | A | n-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4ll5 | A | A | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4ll5 | A | B | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4lm5 | A | A | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4lm5 | A | B | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4lmu | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4lmu | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4mbi | A | n,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4mbl | A | (1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4mta | A | 2-methyl-5-phenylfuran-3-carboxylic acid | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4n6y | A | 2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4n6z | A | 3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4n70 | A | A | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4n70 | A | B | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4rbl | A | 1,4,5,8-tetrahydroxyanthracene-9,10-dione | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4rc2 | A | 1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dione | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4rc3 | A | 1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dione | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4rc4 | A | 1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dione | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4rpv | A | (3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4ty1 | A | n-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4wrs | A | 3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazole | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4wsy | A | 5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4wt6 | A | 6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4xh6 | A | 5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 4xhk | B | A | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 4xhk | B | B | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5c1q | B | 3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-one | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5dgz | A | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5dhj | A | A | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5dhj | A | B | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | Show | ![]() |
![]() | PIM1 | PIM | CAMK | 5dia | A | (1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamine | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5dwr | A | n-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | Show | ![]() | |
![]() | PIM1 | PIM | CAMK | 5eol | A | macrocyclic quinoxaline-pyrrolodihydropiperidinone | Human | Show | ![]() |


