Browse kinase entries (page 230 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PIM1PIMCAMK4as0ABphtalimide-ruthenium complexHumanShow
PIM1PIMCAMK4bznAn-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHumanShow
PIM1PIMCAMK4bzoAn-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHumanShow
PIM1PIMCAMK4dtkAA(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHumanShow
PIM1PIMCAMK4dtkAB(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHumanShow
PIM1PIMCAMK4enxA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-oneHumanShow
PIM1PIMCAMK4enyAA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHumanShow
PIM1PIMCAMK4enyAB(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHumanShow
PIM1PIMCAMK4gw8AA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
PIM1PIMCAMK4gw8AB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
PIM1PIMCAMK4i41A1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedioneHumanShow
PIM1PIMCAMK4iaaA10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazineHumanShow
PIM1PIMCAMK4jx3A-HumanShow
PIM1PIMCAMK4jx7A2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-oneHumanShow
PIM1PIMCAMK4k0yAAn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHumanShow
PIM1PIMCAMK4k0yABn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHumanShow
PIM1PIMCAMK4k18A5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamideHumanShow
PIM1PIMCAMK4k1bAn-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHumanShow
PIM1PIMCAMK4ll5AA6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHumanShow
PIM1PIMCAMK4ll5AB6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHumanShow
PIM1PIMCAMK4lm5AA2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHumanShow
PIM1PIMCAMK4lm5AB2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHumanShow
PIM1PIMCAMK4lmuAA3,5,7,3',4'-pentahydroxyflavoneHumanShow
PIM1PIMCAMK4lmuAB3,5,7,3',4'-pentahydroxyflavoneHumanShow
PIM1PIMCAMK4mbiAn,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamineHumanShow
PIM1PIMCAMK4mblA(1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamineHumanShow
PIM1PIMCAMK4mtaA2-methyl-5-phenylfuran-3-carboxylic acidHumanShow
PIM1PIMCAMK4n6yA2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHumanShow
PIM1PIMCAMK4n6zA3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamideHumanShow
PIM1PIMCAMK4n70AAn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHumanShow
PIM1PIMCAMK4n70ABn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHumanShow
PIM1PIMCAMK4rblA1,4,5,8-tetrahydroxyanthracene-9,10-dioneHumanShow
PIM1PIMCAMK4rc2A1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dioneHumanShow
PIM1PIMCAMK4rc3A1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dioneHumanShow
PIM1PIMCAMK4rc4A1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dioneHumanShow
PIM1PIMCAMK4rpvA(3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amineHumanShow
PIM1PIMCAMK4ty1An-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amineHumanShow
PIM1PIMCAMK4wrsA3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazoleHumanShow
PIM1PIMCAMK4wsyA5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amineHumanShow
PIM1PIMCAMK4wt6A6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amineHumanShow
PIM1PIMCAMK4xh6A5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-oneHumanShow
PIM1PIMCAMK4xhkBA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHumanShow
PIM1PIMCAMK4xhkBB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHumanShow
PIM1PIMCAMK5c1qB3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-oneHumanShow
PIM1PIMCAMK5dgzA(2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amineHumanShow
PIM1PIMCAMK5dhjAA3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHumanShow
PIM1PIMCAMK5dhjAB3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHumanShow
PIM1PIMCAMK5diaA(1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamineHumanShow
PIM1PIMCAMK5dwrAn-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHumanShow
PIM1PIMCAMK5eolA macrocyclic quinoxaline-pyrrolodihydropiperidinoneHumanShow
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