Browse kinase entries (page 25 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
BRAFRAFTKL6n0qBAn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHumanShow
BRAFRAFTKL6n0qBBn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHumanShow
BRAFRAFTKL6nsqA5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHumanShow
BRAFRAFTKL6nsqB5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHumanShow
BRAFRAFTKL6nybAphosphothiophosphoric acid-adenylate esterHumanShow
BRAFRAFTKL6p3dA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
BRAFRAFTKL6p7gA3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHumanShow
BRAFRAFTKL6p7gB3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHumanShow
BRAFRAFTKL6p7gC3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHumanShow
BRAFRAFTKL6p7gD3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHumanShow
BRAFRAFTKL6pp9AAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL6pp9ABphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL6q0jAA-HumanShow
BRAFRAFTKL6q0jAB-HumanShow
BRAFRAFTKL6q0jBA-HumanShow
BRAFRAFTKL6q0jBB-HumanShow
BRAFRAFTKL6q0kA-HumanShow
BRAFRAFTKL6q0kB-HumanShow
BRAFRAFTKL6q0tAA-HumanShow
BRAFRAFTKL6q0tAB-HumanShow
BRAFRAFTKL6q0tBA-HumanShow
BRAFRAFTKL6q0tBB-HumanShow
BRAFRAFTKL6u2gBphosphomethylphosphonic acid adenylate esterHumanShow
BRAFRAFTKL6u2hCA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHumanShow
BRAFRAFTKL6u2hDA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHumanShow
BRAFRAFTKL6uanB-HumanShow
BRAFRAFTKL6uanC-HumanShow
BRAFRAFTKL6uuoA1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHumanShow
BRAFRAFTKL6uuoB1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHumanShow
BRAFRAFTKL6v2uAdabrafenibHumanShow
BRAFRAFTKL6v2uBdabrafenibHumanShow
BRAFRAFTKL6v2wAAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL6v2wABphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL6v34A6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHumanShow
BRAFRAFTKL6v34B6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHumanShow
BRAFRAFTKL6xagCA-HumanShow
BRAFRAFTKL6xagDA-HumanShow
BRAFRAFTKL6xfpAA4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamideHumanShow
BRAFRAFTKL6xfpAB4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamideHumanShow
BRAFRAFTKL6xloA3-(2-cyanopropan-2-yl)-n-[2-fluoro-4-methyl-5-(7-methyl-8-oxo-7,8-dihydropyrido[2,3-d]pyridazin-3-yl)phenyl]benzamideHumanShow
BRAFRAFTKL7k0vAAn-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}ureaHumanShow
BRAFRAFTKL7k0vABn-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}ureaHumanShow
BRAFRAFTKL7m0tAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0uAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0vAAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0vABphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0wAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0xAAphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0xABphosphoaminophosphonic acid-adenylate esterHumanShow
BRAFRAFTKL7m0yAphosphoaminophosphonic acid-adenylate esterHumanShow
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