Browse kinase entries (page 247 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
RIPK1RIPKTKL5hx6B5-benzyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1,2-oxazole-3-carboxamideHumanShow
RIPK1RIPKTKL5tx5AAgsk2982772HumanShow
RIPK1RIPKTKL5tx5ABgsk2982772HumanShow
RIPK1RIPKTKL5tx5BAgsk2982772HumanShow
RIPK1RIPKTKL5tx5BBgsk2982772HumanShow
RIPK1RIPKTKL6c3eAA2-benzyl-5-nitro-1h-benzimidazoleHumanShow
RIPK1RIPKTKL6c3eAB2-benzyl-5-nitro-1h-benzimidazoleHumanShow
RIPK1RIPKTKL6c3eBA2-benzyl-5-nitro-1h-benzimidazoleHumanShow
RIPK1RIPKTKL6c3eBB2-benzyl-5-nitro-1h-benzimidazoleHumanShow
RIPK1RIPKTKL6c4dA(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHumanShow
RIPK1RIPKTKL6c4dB(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHumanShow
RIPK1RIPKTKL6c4dC(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHumanShow
RIPK1RIPKTKL6c4dD(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHumanShow
RIPK1RIPKTKL6hhoA6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrileHumanShow
RIPK1RIPKTKL6hhoB6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrileHumanShow
RIPK1RIPKTKL6nw2AA(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHumanShow
RIPK1RIPKTKL6nw2AB(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHumanShow
RIPK1RIPKTKL6nw2BA(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHumanShow
RIPK1RIPKTKL6nw2BB(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHumanShow
RIPK1RIPKTKL6nyhA(5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamideHumanShow
RIPK1RIPKTKL6nyhB(5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamideHumanShow
RIPK1RIPKTKL6ocqAA1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHumanShow
RIPK1RIPKTKL6ocqAB1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHumanShow
RIPK1RIPKTKL6ocqBA1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHumanShow
RIPK1RIPKTKL6ocqBB1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHumanShow
RIPK1RIPKTKL6r5fA[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHumanShow
RIPK1RIPKTKL6r5fB[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHumanShow
RIPK1RIPKTKL6r5fC[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHumanShow
RIPK1RIPKTKL6r5fD[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHumanShow
RIPK1RIPKTKL6rlnA~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamideHumanShow
RIPK1RIPKTKL6rlnB~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamideHumanShow
RIPK1RIPKTKL7fczAn-[(3s)-7-(2-cyclopropylethynyl)-5-methyl-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamideHumanShow
RIPK1RIPKTKL7fd0An-[(3s)-5-methyl-7-[2-(oxan-4-yl)ethynyl]-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamideHumanShow
RIPK1RIPKTKL7xmkA5-[2-(cyclopropylcarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-(3-fluorophenyl)ethyl]-1-methyl-indole-3-carboxamideHumanShow
RIPK1RIPKTKL7ydxAA1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamideHumanShow
RIPK1RIPKTKL7ydxAB1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamideHumanShow
RIPK1RIPKTKL8i2nA~{n}-methyl-1-[4-[[[1-methyl-5-(phenylmethyl)pyrazol-3-yl]carbonylamino]methyl]phenyl]benzimidazole-5-carboxamideHumanShow
RIPK2RIPKTKL4c8bA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
RIPK2RIPKTKL4c8bB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
RIPK2RIPKTKL5ar2AA-HumanShow
RIPK2RIPKTKL5ar2AB-HumanShow
RIPK2RIPKTKL5ar2BA-HumanShow
RIPK2RIPKTKL5ar2BB-HumanShow
RIPK2RIPKTKL5ar3AAphosphomethylphosphonic acid adenylate esterHumanShow
RIPK2RIPKTKL5ar3ABphosphomethylphosphonic acid adenylate esterHumanShow
RIPK2RIPKTKL5ar3BAphosphomethylphosphonic acid adenylate esterHumanShow
RIPK2RIPKTKL5ar3BBphosphomethylphosphonic acid adenylate esterHumanShow
RIPK2RIPKTKL5ar4A4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHumanShow
RIPK2RIPKTKL5ar4B4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHumanShow
RIPK2RIPKTKL5ar5AA2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamideHumanShow
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