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Updated: 01-Nov-2025

Browse kinase entries (page 250 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
ROCK1DMPKAGC3d9vA(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazineHumanShow
ROCK1DMPKAGC3d9vB(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazineHumanShow
ROCK1DMPKAGC3nczAcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHumanShow
ROCK1DMPKAGC3nczBcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHumanShow
ROCK1DMPKAGC3nczCcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHumanShow
ROCK1DMPKAGC3nczDcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHumanShow
ROCK1DMPKAGC3ndmA-HumanShow
ROCK1DMPKAGC3ndmB(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHumanShow
ROCK1DMPKAGC3ndmC(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHumanShow
ROCK1DMPKAGC3ndmD(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHumanShow
ROCK1DMPKAGC3tv7A1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3tv7B1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3tv7C1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3tv7D1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3twjA1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3twjB-HumanShow
ROCK1DMPKAGC3twjC1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHumanShow
ROCK1DMPKAGC3twjD-HumanShow
ROCK1DMPKAGC3v8sA1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHumanShow
ROCK1DMPKAGC3v8sB1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHumanShow
ROCK1DMPKAGC3v8sC1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHumanShow
ROCK1DMPKAGC3v8sD1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHumanShow
ROCK1DMPKAGC4w7pAn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHumanShow
ROCK1DMPKAGC4w7pBn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHumanShow
ROCK1DMPKAGC4w7pCn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHumanShow
ROCK1DMPKAGC4w7pDn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHumanShow
ROCK1DMPKAGC4yvcA2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamideHumanShow
ROCK1DMPKAGC4yvcB2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamideHumanShow
ROCK1DMPKAGC4yveA2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHumanShow
ROCK1DMPKAGC4yveB2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHumanShow
ROCK1DMPKAGC5bmlAn-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamideHumanShow
ROCK1DMPKAGC5bmlBn-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamideHumanShow
ROCK1DMPKAGC5hvuA2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHumanShow
ROCK1DMPKAGC5hvuB2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHumanShow
ROCK1DMPKAGC5kksA2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHumanShow
ROCK1DMPKAGC5kksB2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHumanShow
ROCK1DMPKAGC5kktA2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHumanShow
ROCK1DMPKAGC5kktB2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHumanShow
ROCK1DMPKAGC5uzjAn-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamideHumanShow
ROCK1DMPKAGC5uzjBn-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamideHumanShow
ROCK1DMPKAGC5wneA3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHumanShow
ROCK1DMPKAGC5wneB3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHumanShow
ROCK1DMPKAGC5wneC3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHumanShow
ROCK1DMPKAGC5wneD3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHumanShow
ROCK1DMPKAGC5wnfAA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
ROCK1DMPKAGC5wnfAB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
ROCK1DMPKAGC5wnfBA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
ROCK1DMPKAGC5wnfBB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
ROCK1DMPKAGC5wnfCA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
ROCK1DMPKAGC5wnfCB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHumanShow
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