PDB-code
Browse kinase entries (page 253 of 282)
First 249 250 251 PreviousLast257 256 255 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | RPS6KA2 (RSK1) | RSK | AGC | 8xov | A | phosphoaminophosphonic acid-adenylate ester | Human | Show |  | |
| RPS6KA2-b (RSK1-b) | RSKb | CAMK | 8wf4 | A | - | Human | Show | | |
| Rps6ka3 (RSK2) | RSK | AGC | 3g51 | A | phosphoaminophosphonic acid-adenylate ester | Mouse | Show | | |
| Rps6ka3 (RSK2) | RSK | AGC | 3ubd | A | A | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranoside | Mouse | Show | |
| Rps6ka3 (RSK2) | RSK | AGC | 3ubd | A | B | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranoside | Mouse | Show | |
| Rps6ka3 (RSK2) | RSK | AGC | 4el9 | A | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | Show | | |
| Rps6ka3 (RSK2) | RSK | AGC | 4gue | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | Show | |
| Rps6ka3 (RSK2) | RSK | AGC | 4gue | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | A | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | B | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | A | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | B | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | A | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | B | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | Show | | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | A | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | B | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 7opo | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | Show | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | Show | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | A | - | Mouse | Show | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | B | - | Mouse | Show | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | A | - | Mouse | Show | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | B | - | Mouse | Show | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4m8t | A | (2e)-2-cyano-3-[3-(1h-pyrazol-4-yl)phenyl]prop-2-enamide | Mouse | Show | | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4mao | A | (2z)-2-(1h-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]prop-2-enenitrile | Mouse | Show | | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 5o1s | A | dimethyl fumarate | Mouse | Show | | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9t | A | methyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoate | Human | Show | | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9u | A | tert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoate | Human | Show | | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg6 | A | (2s)-2-cyano-3-(1h-indazol-5-yl)propanamide | Human | Show | | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | A | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | Show | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | B | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | Show | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | Show | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | Show | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 8xey | A | - | Human | Show | | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | A | - | Human | Show | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | B | - | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | A | - | Human | Show | | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | B | - | Human | Show | | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | A | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | B | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | A | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | B | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | A | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | B | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | Show | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | Show | |
