PDB-code
Browse kinase entries (page 267 of 282)
First 263 264 265 PreviousLast271 270 269 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | TNIK | STE20 | STE | 2x7f | A | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | A | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | B | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | B | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | C | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | C | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | D | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | D | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | E | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 2x7f | E | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 5ax9 | A | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5ax9 | B | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5ax9 | C | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5cwz | A | - | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5cwz | B | - | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5cwz | C | - | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5d7a | A | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5d7a | B | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 5d7a | C | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 6ra5 | A | 5-bromanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-8-amine | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 6ra5 | B | - | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 6ra7 | A | A | 2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-ol | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 6ra7 | A | B | 2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-ol | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 7xzq | A | - | Human | Show | ![]() | |
![]() | TNIK | STE20 | STE | 7xzr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 7xzr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 8wm0 | A | A | adenosine | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 8wm0 | A | B | adenosine | Human | Show | ![]() |
![]() | TNIK | STE20 | STE | 8x88 | A | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u46 | A | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u46 | B | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u4d | A | debromohymenialdisine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u4d | B | debromohymenialdisine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u54 | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 1u54 | B | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 3eqp | A | n-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 3eqp | B | n-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 3eqr | A | n~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 3eqr | B | n~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4ewh | A | 6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4ewh | B | 6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4hzr | A | A | - | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 4hzr | A | B | - | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 4hzr | B | A | - | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 4hzr | B | B | - | Human | Show | ![]() |
![]() | TNK2 (ACK) | Ack | TK | 4hzs | A | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4hzs | B | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4hzs | C | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4hzs | D | - | Human | Show | ![]() | |
![]() | TNK2 (ACK) | Ack | TK | 4id7 | A | cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol | Human | Show | ![]() |


