PDB-code
Browse kinase entries (page 270 of 282)
First 266 267 268 PreviousLast274 273 272 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | TTK | TTK | Other | 2zmc | A | - | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 2zmd | A | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3cek | A | - | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3dbq | A | - | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3gfw | A | 1-(4-(4-(2-(isopropylsulfonyl)phenylamino)-1h-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-ol | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3h9f | A | A | 9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-one | Human | Show | ![]() |
![]() | TTK | TTK | Other | 3h9f | A | B | 9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-one | Human | Show | ![]() |
![]() | TTK | TTK | Other | 3hmn | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3hmo | A | staurosporine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3hmp | A | 7-chloro-n-(cyclopropylmethyl)quinazolin-4-amine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3vqu | A | 4-[(4-amino-5-cyano-6-ethoxypyridin-2-yl)amino]benzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3w1f | A | 5-[5-ethoxy-6-(1-methyl-1h-pyrazol-4-yl)-1h-indazol-3-yl]-2-methylbenzenesulfonamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3wyx | A | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3wyy | A | (2e)-3-[4-({4-amino-5-cyano-6-[(3s,5s,7s)-tricyclo[3.3.1.1~3,7~]dec-1-ylamino]pyridin-2-yl}amino)-2-(cyanomethoxy)phenyl]-n-(2-methoxyethyl)prop-2-enamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3wzj | A | 4-{6-(cyclohexylamino)-8-[(tetrahydro-2h-pyran-4-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-n-cyclopropylbenzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 3wzk | A | n-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4bhz | A | thieno[2,3-c][2,6]naphthyridine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4bi0 | A | 5h-pyrimido[5,4-b]indole | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4bi1 | A | thieno[3,2-c][2,6]naphthyridine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4bi2 | A | thieno[2,3-c][2,7]naphthyridine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4c4e | A | A | n-(3,4-dimethoxyphenyl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | Show | ![]() |
![]() | TTK | TTK | Other | 4c4e | A | B | - | Human | Show | ![]() |
![]() | TTK | TTK | Other | 4c4f | A | n-(2-methoxyphenyl)-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4c4g | A | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4c4h | A | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4c4i | A | tert-butyl 6-{[2-chloro-4-(dimethylcarbamoyl)phenyl]amino}-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4c4j | A | tert-butyl 6-{[2-chloro-4-(1-methyl-1h-imidazol-5-yl)phenyl]amino}-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4cv8 | A | 3-amino-5-(1-methyl-1h-pyrazol-4-yl)pyridin-2(1h)-one | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4cv9 | A | 4-(4-methylpiperazin-1-yl)-n-(2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin-3-yl)benzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4cva | A | n-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)-4-(piperidin-1-yl)benzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4d2s | A | n-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4js8 | A | 4-(cyclohexylmethoxy)-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-2h-indazole | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4jt3 | A | 2-phenyl-n-[3-(3-sulfamoylphenyl)-2h-indazol-5-yl]acetamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4o6l | A | n-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4o6l | B | n-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 4zeg | A | n-cyclopropyl-2-methyl-4-(7-{[2-(morpholin-4-yl)ethyl]amino}-5-phenoxypyrazolo[1,5-a]pyrimidin-3-yl)benzamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap0 | A | 9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-one | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap1 | A | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap2 | A | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap3 | A | 9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-one | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap4 | A | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap5 | A | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ap6 | A | A | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() |
![]() | TTK | TTK | Other | 5ap6 | A | B | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | Show | ![]() |
![]() | TTK | TTK | Other | 5ap7 | A | n-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5eh0 | A | n2-(2-methoxy-4-(1-methyl-1h-pyrazol-4-yl)phenyl)-n8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ehl | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5eho | A | ~{n}8-cyclohexyl-~{n}2-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ehy | A | 4-(furan-3-yl)-3-phenyl-2~{h}-pyrazolo[4,3-c]pyridine | Human | Show | ![]() | |
![]() | TTK | TTK | Other | 5ei2 | A | ~{n}-(2,4-dimethoxyphenyl)-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine | Human | Show | ![]() |


