Browse kinase entries (page 279 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
VRK2VRKCK16ncgB4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHumanShow
VRK2VRKCK18q1zAA2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHumanShow
VRK2VRKCK18q1zAB2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHumanShow
VRK3VRKCK12jiiAA-HumanShow
VRK3VRKCK12jiiAB-HumanShow
VRK3VRKCK12jiiBA-HumanShow
VRK3VRKCK12jiiBB-HumanShow
WEE1 (Wee1)WEEOther1x8bA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther2in6A3-(9-hydroxy-1,3-dioxo-4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-6(1h)-yl)propanoic acidHumanShow
WEE1 (Wee1)WEEOther2io6A9-hydroxy-6-(3-hydroxypropyl)-4-(2-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther2z2wAn-[4-(2-chlorophenyl)-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-9-yl]formamideHumanShow
WEE1 (Wee1)WEEOther3bi6AA4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamideHumanShow
WEE1 (Wee1)WEEOther3bi6AB4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamideHumanShow
WEE1 (Wee1)WEEOther3bizAA4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther3bizAB4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther3cqeAA8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamideHumanShow
WEE1 (Wee1)WEEOther3cqeAB8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamideHumanShow
WEE1 (Wee1)WEEOther3cr0AA4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther3cr0AB4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dioneHumanShow
WEE1 (Wee1)WEEOther5v5yA1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vc3A4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
WEE1 (Wee1)WEEOther5vc4A4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
WEE1 (Wee1)WEEOther5vc5AA6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
WEE1 (Wee1)WEEOther5vc5AB6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHumanShow
WEE1 (Wee1)WEEOther5vc6An,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
WEE1 (Wee1)WEEOther5vd2An-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHumanShow
WEE1 (Wee1)WEEOther5vd4A6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1-{6-[(1s)-2,2,2-trifluoro-1-hydroxyethyl]pyridin-2-yl}-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vd5A1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(morpholin-4-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vd7A6-{[3-fluoro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vd8A6-{[3-chloro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vd9A1-{6-[(1r)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther5vdaA1-{6-[(1s)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther7n3uA1-[(7r)-7-ethyl-7-hydroxy-7h-cyclopenta[b]pyridin-2-yl]-6-[4-(4-methylpiperazin-1-yl)anilino]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther8bjuAA2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE1 (Wee1)WEEOther8bjuAB2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WEE2 (Wee1B)WEEOther5vdkA1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHumanShow
WNK1 (Wnk1)WNKOther4pwnA-HumanShow
WNK1 (Wnk1)WNKOther5tf9A{2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanoneHumanShow
WNK1 (Wnk1)WNKOther5tf9B{2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanoneHumanShow
WNK1 (Wnk1)WNKOther5wdyAAphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5wdyABphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5wdyBAphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5wdyBBphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5we8AAphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5we8ABphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5we8BAphosphoaminophosphonic acid-adenylate esterHumanShow
WNK1 (Wnk1)WNKOther5we8BBphosphoaminophosphonic acid-adenylate esterHumanShow
WNK3 (Wnk3)WNKOther5o1vAA-HumanShow
WNK3 (Wnk3)WNKOther5o1vAB-HumanShow
WNK3 (Wnk3)WNKOther5o1vBA-HumanShow
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