PDB-code
Browse kinase entries (page 35 of 282)
First 31 32 33 PreviousLast39 38 37 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CASK | CASK | CAMK | 7oal | A | 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | A | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | B | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 3tku | A | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 3tku | B | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | A | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | B | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 5ote | A | 2-[4-[(6~{s})-1,8-diazaspiro[5.5]undecan-8-yl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-1,3-thiazole | Human | Show | ![]() | |
![]() | CDC42BPB (MRCKb) | DMPK | AGC | 5otf | A | (6~{s})-8-(3-pyrimidin-4-yl-1~{h}-pyrrolo[2,3-b]pyridin-4-yl)-1,8-diazaspiro[5.5]undecane | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f99 | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f9a | A | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f9a | C | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f9b | A | 2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f9b | C | 2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 4f9c | A | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | Show | ![]() | |
![]() | CDC7 | CDC7 | Other | 6ya6 | A | A | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | Show | ![]() |
![]() | CDC7 | CDC7 | Other | 6ya6 | A | B | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | Show | ![]() |
![]() | CDC7 | CDC7 | Other | 6ya7 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDC7 | CDC7 | Other | 6ya7 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDC7 | CDC7 | Other | 6ya8 | A | A | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDC7 | CDC7 | Other | 6ya8 | A | B | adenosine-5'-diphosphate | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4y72 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4y72 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | A | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | B | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | A | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | B | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | A | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | B | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | A | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | B | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | A | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | B | - | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5lqf | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5lqf | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5lqf | D | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 5lqf | D | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | A | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | B | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | Show | ![]() |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu3 | A | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu4 | A | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu6 | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu7 | A | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu7 | C | - | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu7 | E | - | Human | Show | ![]() | |
![]() | CDK1 (CDC2) | CDK | CMGC | 6gu7 | G | - | Human | Show | ![]() |


