Browse kinase entries (page 37 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK13 (CHED)CDKCMGC7nxjAn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHumanShow
CDK16 (PCTAIRE1)CDKCMGC3mtlAA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}HumanShow
CDK16 (PCTAIRE1)CDKCMGC3mtlAB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}HumanShow
CDK16 (PCTAIRE1)CDKCMGC5g6vA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
CDK16 (PCTAIRE1)CDKCMGC5g6vB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
CDK2CDKCMGC1aq1AstaurosporineHumanShow
CDK2CDKCMGC1b38Aadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1b39Aadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1buhA-HumanShow
CDK2CDKCMGC1ckpAApurvalanol bHumanShow
CDK2CDKCMGC1ckpABpurvalanol bHumanShow
CDK2CDKCMGC1di8A4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHumanShow
CDK2CDKCMGC1dm2AA4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHumanShow
CDK2CDKCMGC1dm2AB4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHumanShow
CDK2CDKCMGC1e1vA6-o-cyclohexylmethyl guanineHumanShow
CDK2CDKCMGC1e1xA6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamineHumanShow
CDK2CDKCMGC1e9hA2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHumanShow
CDK2CDKCMGC1e9hC2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHumanShow
CDK2CDKCMGC1f5qAA-HumanShow
CDK2CDKCMGC1f5qAB-HumanShow
CDK2CDKCMGC1f5qCA-HumanShow
CDK2CDKCMGC1f5qCB-HumanShow
CDK2CDKCMGC1finAadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1finCadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1fq1Badenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1fvtA4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamideHumanShow
CDK2CDKCMGC1fvvA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHumanShow
CDK2CDKCMGC1fvvC4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHumanShow
CDK2CDKCMGC1g5sA2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurineHumanShow
CDK2CDKCMGC1gihA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHumanShow
CDK2CDKCMGC1giiA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHumanShow
CDK2CDKCMGC1gijA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-ureaHumanShow
CDK2CDKCMGC1gy3Aadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1gy3Cadenosine-5'-triphosphateHumanShow
CDK2CDKCMGC1gz8AA1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHumanShow
CDK2CDKCMGC1gz8AB1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHumanShow
CDK2CDKCMGC1h00AA(2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h00AB(2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h01AA(2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h01AB(2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h07AA((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHumanShow
CDK2CDKCMGC1h07AB((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHumanShow
CDK2CDKCMGC1h08AA(2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h08AB(2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHumanShow
CDK2CDKCMGC1h0vAA5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHumanShow
CDK2CDKCMGC1h0vAB5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHumanShow
CDK2CDKCMGC1h0wAA1-amino-6-cyclohex-3-enylmethyloxypurineHumanShow
CDK2CDKCMGC1h0wAB1-amino-6-cyclohex-3-enylmethyloxypurineHumanShow
CDK2CDKCMGC1h1pA6-o-cyclohexylmethyl guanineHumanShow
CDK2CDKCMGC1h1pC6-o-cyclohexylmethyl guanineHumanShow
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