PDB-code
Browse kinase entries (page 37 of 282)
First 33 34 35 PreviousLast41 40 39 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | CDK13 (CHED) | CDK | CMGC | 7nxj | A | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | Show | ![]() | |
![]() | CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | ![]() |
![]() | CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | Show | ![]() |
![]() | CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | ![]() | |
![]() | CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1aq1 | A | staurosporine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1b38 | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1b39 | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1buh | A | - | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1ckp | A | A | purvalanol b | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1ckp | A | B | purvalanol b | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1di8 | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1dm2 | A | A | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1dm2 | A | B | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1e1v | A | 6-o-cyclohexylmethyl guanine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1e1x | A | 6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1e9h | A | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1e9h | C | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1f5q | A | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1f5q | A | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1f5q | C | A | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1f5q | C | B | - | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1fin | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1fin | C | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1fq1 | B | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1fvt | A | 4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1fvv | A | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1fvv | C | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1g5s | A | 2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gih | A | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gii | A | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gij | A | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-urea | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gy3 | A | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gy3 | C | adenosine-5'-triphosphate | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1gz8 | A | A | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1gz8 | A | B | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h00 | A | A | (2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h00 | A | B | (2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h01 | A | A | (2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h01 | A | B | (2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h07 | A | A | ((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h07 | A | B | ((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h08 | A | A | (2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h08 | A | B | (2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h0v | A | A | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h0v | A | B | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h0w | A | A | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h0w | A | B | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | Show | ![]() |
![]() | CDK2 | CDK | CMGC | 1h1p | A | 6-o-cyclohexylmethyl guanine | Human | Show | ![]() | |
![]() | CDK2 | CDK | CMGC | 1h1p | C | 6-o-cyclohexylmethyl guanine | Human | Show | ![]() |


