Browse kinase entries (page 42 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC2r3jAB3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3kAA3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHumanShow
CDK2CDKCMGC2r3kAB3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHumanShow
CDK2CDKCMGC2r3kAC3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHumanShow
CDK2CDKCMGC2r3lAA3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHumanShow
CDK2CDKCMGC2r3lAB3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHumanShow
CDK2CDKCMGC2r3lAC3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHumanShow
CDK2CDKCMGC2r3mAAn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3mABn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3nAA3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3nAB3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3oAA(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHumanShow
CDK2CDKCMGC2r3oAB(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHumanShow
CDK2CDKCMGC2r3oAC(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHumanShow
CDK2CDKCMGC2r3pAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3pAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3qAA3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHumanShow
CDK2CDKCMGC2r3qAB3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHumanShow
CDK2CDKCMGC2r3qAC3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHumanShow
CDK2CDKCMGC2r3rAA3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r3rAB3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHumanShow
CDK2CDKCMGC2r64An-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamideHumanShow
CDK2CDKCMGC2uueA4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHumanShow
CDK2CDKCMGC2uueC4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHumanShow
CDK2CDKCMGC2uzbAC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC2uzbAD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC2uzbCC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC2uzbCD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC2uzdA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHumanShow
CDK2CDKCMGC2uzdC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHumanShow
CDK2CDKCMGC2uzeA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHumanShow
CDK2CDKCMGC2uzeC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHumanShow
CDK2CDKCMGC2uzlA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHumanShow
CDK2CDKCMGC2uzlC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHumanShow
CDK2CDKCMGC2uznA4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamideHumanShow
CDK2CDKCMGC2uzoA4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHumanShow
CDK2CDKCMGC2v0dA2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-oneHumanShow
CDK2CDKCMGC2v22A-HumanShow
CDK2CDKCMGC2v22C-HumanShow
CDK2CDKCMGC2vtaA1h-indazoleHumanShow
CDK2CDKCMGC2vthA5-hydroxynaphthalene-1-sulfonamideHumanShow
CDK2CDKCMGC2vtiAn-(4-sulfamoylphenyl)-1h-indazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtjA4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamideHumanShow
CDK2CDKCMGC2vtlAn-phenyl-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtmApyrazolo[1,5-a]pyrimidine-3-carbonitrileHumanShow
CDK2CDKCMGC2vtnA4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtoAAn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtoABn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtpAA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtpAB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHumanShow
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