Browse kinase entries (page 43 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC2vtqA{[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vtrAA5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHumanShow
CDK2CDKCMGC2vtrAB5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHumanShow
CDK2CDKCMGC2vtsA5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHumanShow
CDK2CDKCMGC2vttA4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vu3AA4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vu3AB4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHumanShow
CDK2CDKCMGC2vv9AA2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHumanShow
CDK2CDKCMGC2vv9AB2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHumanShow
CDK2CDKCMGC2w05AAn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHumanShow
CDK2CDKCMGC2w05ABn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHumanShow
CDK2CDKCMGC2w06A4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC2w17AAn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2w17ABn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHumanShow
CDK2CDKCMGC2w1hAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHumanShow
CDK2CDKCMGC2wevAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wevAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wevAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wevCA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wevCB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wevCC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHumanShow
CDK2CDKCMGC2wfyAA-HumanShow
CDK2CDKCMGC2wfyAB-HumanShow
CDK2CDKCMGC2wfyCA-HumanShow
CDK2CDKCMGC2wfyCB-HumanShow
CDK2CDKCMGC2whbAA-HumanShow
CDK2CDKCMGC2whbAB-HumanShow
CDK2CDKCMGC2whbCA-HumanShow
CDK2CDKCMGC2whbCB-HumanShow
CDK2CDKCMGC2wihAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
CDK2CDKCMGC2wihCn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
CDK2CDKCMGC2wipA1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHumanShow
CDK2CDKCMGC2wipC1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHumanShow
CDK2CDKCMGC2wmaA-HumanShow
CDK2CDKCMGC2wmaC-HumanShow
CDK2CDKCMGC2wmbA-HumanShow
CDK2CDKCMGC2wmbC-HumanShow
CDK2CDKCMGC2wpaAn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHumanShow
CDK2CDKCMGC2wpaCn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHumanShow
CDK2CDKCMGC2wxvAn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
CDK2CDKCMGC2wxvCn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHumanShow
CDK2CDKCMGC2x1nAA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHumanShow
CDK2CDKCMGC2x1nAB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHumanShow
CDK2CDKCMGC2x1nCA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHumanShow
CDK2CDKCMGC2x1nCB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHumanShow
CDK2CDKCMGC2xmyAA4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHumanShow
CDK2CDKCMGC2xmyAB4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHumanShow
CDK2CDKCMGC2xnbAA3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHumanShow
CDK2CDKCMGC2xnbAB3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHumanShow
CDK2CDKCMGC3bhtAA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
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