Browse kinase entries (page 48 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC3rzbAB4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHumanShow
CDK2CDKCMGC3s00AA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHumanShow
CDK2CDKCMGC3s00AB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHumanShow
CDK2CDKCMGC3s0oAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHumanShow
CDK2CDKCMGC3s0oAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHumanShow
CDK2CDKCMGC3s1hAA4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC3s1hAB4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC3s2pA(3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diolHumanShow
CDK2CDKCMGC3sqqAA4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC3sqqAB4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHumanShow
CDK2CDKCMGC3sw4AAn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHumanShow
CDK2CDKCMGC3sw4ABn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHumanShow
CDK2CDKCMGC3sw7AAn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHumanShow
CDK2CDKCMGC3sw7ABn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHumanShow
CDK2CDKCMGC3ti1AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHumanShow
CDK2CDKCMGC3ti1ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHumanShow
CDK2CDKCMGC3tiyAA2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHumanShow
CDK2CDKCMGC3tiyAB2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHumanShow
CDK2CDKCMGC3tizA1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-olHumanShow
CDK2CDKCMGC3tnwAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK2CDKCMGC3tnwAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK2CDKCMGC3tnwCA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK2CDKCMGC3tnwCB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK2CDKCMGC3uliAA1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamideHumanShow
CDK2CDKCMGC3unjA4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHumanShow
CDK2CDKCMGC3unkA4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
CDK2CDKCMGC3wblAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHumanShow
CDK2CDKCMGC4acmAA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHumanShow
CDK2CDKCMGC4acmAB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHumanShow
CDK2CDKCMGC4bckAA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckAB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckAC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckAD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckCA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckCB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckCC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bckCD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK2CDKCMGC4bcmAA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcmAB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcmCA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcmCB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcnAA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcnAB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcnCA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcnCB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcoAA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcoAB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcoCA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcoCB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcpAA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
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