Browse kinase entries (page 49 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK2CDKCMGC4bcpAB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcpCA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcpCB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcqAA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcqAB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcqCA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bcqCB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHumanShow
CDK2CDKCMGC4bghAA4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHumanShow
CDK2CDKCMGC4bghAB4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHumanShow
CDK2CDKCMGC4bzdAA6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHumanShow
CDK2CDKCMGC4bzdAB6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHumanShow
CDK2CDKCMGC4cfmAA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfmAB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfmCA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfmCB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfnAA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfnAB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfnCA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfnCB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHumanShow
CDK2CDKCMGC4cfuAA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHumanShow
CDK2CDKCMGC4cfuAB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHumanShow
CDK2CDKCMGC4cfuCA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHumanShow
CDK2CDKCMGC4cfuCB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHumanShow
CDK2CDKCMGC4cfvAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHumanShow
CDK2CDKCMGC4cfvAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHumanShow
CDK2CDKCMGC4cfvCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHumanShow
CDK2CDKCMGC4cfvCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHumanShow
CDK2CDKCMGC4cfwAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfwAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfwAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfwCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfwCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfwCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHumanShow
CDK2CDKCMGC4cfxAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4cfxAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4cfxAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4cfxCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4cfxCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4cfxCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHumanShow
CDK2CDKCMGC4d1xA(4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHumanShow
CDK2CDKCMGC4d1zA(4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHumanShow
CDK2CDKCMGC4ek3AA-HumanShow
CDK2CDKCMGC4ek3AB-HumanShow
CDK2CDKCMGC4ek4AA4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHumanShow
CDK2CDKCMGC4ek4AB4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHumanShow
CDK2CDKCMGC4ek4AC4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHumanShow
CDK2CDKCMGC4ek5AAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHumanShow
CDK2CDKCMGC4ek5ABn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHumanShow
CDK2CDKCMGC4ek6AAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHumanShow
CDK2CDKCMGC4ek6ABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHumanShow
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