Browse kinase entries (page 58 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK8CDKCMGC5idpAA(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHumanShow
CDK8CDKCMGC5idpAB(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHumanShow
CDK8CDKCMGC5xqxAn-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHumanShow
CDK8CDKCMGC5xs2AA3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHumanShow
CDK8CDKCMGC5xs2AB3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHumanShow
CDK8CDKCMGC6qtgA2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamideHumanShow
CDK8CDKCMGC6qtjA~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamideHumanShow
CDK8CDKCMGC6r3sAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHumanShow
CDK8CDKCMGC6r3sAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHumanShow
CDK8CDKCMGC6t41A~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amineHumanShow
CDK8CDKCMGC6tpaA1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)ureaHumanShow
CDK8CDKCMGC6y0aAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHumanShow
CDK8CDKCMGC6y0aAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHumanShow
CDK9CDKCMGC3blhA-HumanShow
CDK9CDKCMGC3blqAadenosine-5'-triphosphateHumanShow
CDK9CDKCMGC3blrA2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-oneHumanShow
CDK9CDKCMGC3lq5A(2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHumanShow
CDK9CDKCMGC3mi9A-HumanShow
CDK9CDKCMGC3miaAphosphoaminophosphonic acid-adenylate esterHumanShow
CDK9CDKCMGC3my1A5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHumanShow
CDK9CDKCMGC3tn8A4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK9CDKCMGC3tnhA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHumanShow
CDK9CDKCMGC3tniA-HumanShow
CDK9CDKCMGC4bcfA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK9CDKCMGC4bcgA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK9CDKCMGC4bchA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHumanShow
CDK9CDKCMGC4bciA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHumanShow
CDK9CDKCMGC4bcjA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHumanShow
CDK9CDKCMGC4ec8A-HumanShow
CDK9CDKCMGC4ec9A-HumanShow
CDK9CDKCMGC4imyAAadenosine monophosphateHumanShow
CDK9CDKCMGC4imyABadenosine monophosphateHumanShow
CDK9CDKCMGC4imyCAadenosine monophosphateHumanShow
CDK9CDKCMGC4imyCBadenosine monophosphateHumanShow
CDK9CDKCMGC4imyEAadenosine monophosphateHumanShow
CDK9CDKCMGC4imyEBadenosine monophosphateHumanShow
CDK9CDKCMGC4ogrAadenosineHumanShow
CDK9CDKCMGC4ogrEadenosineHumanShow
CDK9CDKCMGC4ogrIadenosineHumanShow
CDK9CDKCMGC4or5A-HumanShow
CDK9CDKCMGC4or5F-HumanShow
CDK9CDKCMGC5l1zA-HumanShow
CDK9CDKCMGC6cytA-HumanShow
CDK9CDKCMGC6gzhA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHumanShow
CDK9CDKCMGC6w9eAA(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHumanShow
CDK9CDKCMGC6w9eAB(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHumanShow
CDK9CDKCMGC6w9eAC(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHumanShow
CDK9CDKCMGC6w9eAD(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHumanShow
CDK9CDKCMGC6z45A(1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamideHumanShow
CDK9CDKCMGC7nwkAn-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamideHumanShow
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