PDB-code
Browse kinase entries (page 63 of 282)
First 59 60 61 PreviousLast67 66 65 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show |  |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq8 | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | A | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | B | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | A | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | B | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | A | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | B | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | A | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | B | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | A | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | B | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | A | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | B | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | A | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | B | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | A | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | B | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | A | adenine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | B | adenine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | A | n,n-dimethyl-7h-purin-6-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | B | n,n-dimethyl-7h-purin-6-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | B | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjm | A | 4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjo | A | 4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjr | A | 4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | A | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | B | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk1 | A | 4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk2 | A | 4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk3 | A | 4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bkn | A | adenine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bko | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7mck | A | n-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | A | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | B | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | A | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | B | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suh | A | 1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sui | A | (3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suj | A | (3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e80 | A | 2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e81 | A | (1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siv | A | n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siw | A | (1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8six | A | (1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamide | Human | Show | |
