Browse kinase entries (page 93 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DYRK1ADYRKCMGC2vx3CBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2vx3DAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2vx3DBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2wo6AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2wo6ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2wo6BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC2wo6BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHumanShow
DYRK1ADYRKCMGC3anqA(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHumanShow
DYRK1ADYRKCMGC3anqB(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHumanShow
DYRK1ADYRKCMGC3anqC(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHumanShow
DYRK1ADYRKCMGC3anqD(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHumanShow
DYRK1ADYRKCMGC3anrA7-methoxy-1-methyl-9h-beta-carbolineHumanShow
DYRK1ADYRKCMGC3anrB7-methoxy-1-methyl-9h-beta-carbolineHumanShow
DYRK1ADYRKCMGC3anrC7-methoxy-1-methyl-9h-beta-carbolineHumanShow
DYRK1ADYRKCMGC3anrD7-methoxy-1-methyl-9h-beta-carbolineHumanShow
DYRK1ADYRKCMGC4azeA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
DYRK1ADYRKCMGC4azeB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
DYRK1ADYRKCMGC4azeC5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHumanShow
DYRK1ADYRKCMGC4mq1AAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1ABn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1BAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1BBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1CAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1CBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1DAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq1DBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHumanShow
DYRK1ADYRKCMGC4mq2AAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2ABmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2BAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2BBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2CAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2CBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2DAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4mq2DBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHumanShow
DYRK1ADYRKCMGC4nctApkc412HumanShow
DYRK1ADYRKCMGC4nctBpkc412HumanShow
DYRK1ADYRKCMGC4nctCpkc412HumanShow
DYRK1ADYRKCMGC4nctDpkc412HumanShow
DYRK1ADYRKCMGC4yljAA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljAB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljBA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljBB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljCA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljCB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljDA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yljDB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4ylkAA10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4ylkAB10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yllAA10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
DYRK1ADYRKCMGC4yllAB10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHumanShow
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