PDB-code
Browse kinase entries (page 95 of 282)
First 91 92 93 PreviousLast99 98 97 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
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![]() | DYRK1A | DYRK | CMGC | 6eif | B | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eif | C | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eif | D | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eij | A | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eij | B | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eij | C | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eij | D | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eil | A | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eil | B | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eil | C | - | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eil | D | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eip | A | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eip | B | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eip | C | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eip | D | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiq | A | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiq | B | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiq | C | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiq | D | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eir | A | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eir | B | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eir | C | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eir | D | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eis | A | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | A | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | B | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | B | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | C | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | C | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | D | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eis | D | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6eiv | A | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiv | B | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiv | C | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6eiv | D | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6ej4 | A | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6ej4 | B | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6ej4 | C | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6ej4 | D | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6ln1 | A | 1,3,5,8-tetrakis(oxidanyl)xanthen-9-one | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | A | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | A | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | B | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | B | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | C | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | C | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | D | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6qu2 | D | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s11 | A | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s11 | A | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | Show | ![]() |


