Browse kinase entries (page 95 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DYRK1ADYRKCMGC6eifB4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHumanShow
DYRK1ADYRKCMGC6eifC4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHumanShow
DYRK1ADYRKCMGC6eifD4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHumanShow
DYRK1ADYRKCMGC6eijA~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHumanShow
DYRK1ADYRKCMGC6eijB~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHumanShow
DYRK1ADYRKCMGC6eijC~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHumanShow
DYRK1ADYRKCMGC6eijD~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHumanShow
DYRK1ADYRKCMGC6eilA[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHumanShow
DYRK1ADYRKCMGC6eilB[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHumanShow
DYRK1ADYRKCMGC6eilC-HumanShow
DYRK1ADYRKCMGC6eilD[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHumanShow
DYRK1ADYRKCMGC6eipA4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHumanShow
DYRK1ADYRKCMGC6eipB4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHumanShow
DYRK1ADYRKCMGC6eipC4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHumanShow
DYRK1ADYRKCMGC6eipD4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHumanShow
DYRK1ADYRKCMGC6eiqA[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHumanShow
DYRK1ADYRKCMGC6eiqB[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHumanShow
DYRK1ADYRKCMGC6eiqC[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHumanShow
DYRK1ADYRKCMGC6eiqD[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHumanShow
DYRK1ADYRKCMGC6eirA~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eirB~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eirC~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eirD~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eisAA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisAB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisBA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisBB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisCA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisCB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisDA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eisDB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHumanShow
DYRK1ADYRKCMGC6eivA~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eivB~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eivC~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6eivD~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHumanShow
DYRK1ADYRKCMGC6ej4A3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHumanShow
DYRK1ADYRKCMGC6ej4B3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHumanShow
DYRK1ADYRKCMGC6ej4C3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHumanShow
DYRK1ADYRKCMGC6ej4D3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHumanShow
DYRK1ADYRKCMGC6ln1A1,3,5,8-tetrakis(oxidanyl)xanthen-9-oneHumanShow
DYRK1ADYRKCMGC6qu2AA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2AB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2BA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2BB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2CA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2CB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2DA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6qu2DB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHumanShow
DYRK1ADYRKCMGC6s11AA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHumanShow
DYRK1ADYRKCMGC6s11AB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHumanShow
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