Browse kinase entries (page 96 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DYRK1ADYRKCMGC6s11BA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHumanShow
DYRK1ADYRKCMGC6s11BB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHumanShow
DYRK1ADYRKCMGC6s14AA~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s14AB~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s17AA~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s17AB~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1bAA~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1bAB~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1hAA~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1hAB~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iAA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iAB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iBA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iBB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iCA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iCB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iDA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1iDB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC6s1jAA3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHumanShow
DYRK1ADYRKCMGC6s1jAB3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHumanShow
DYRK1ADYRKCMGC6t6aAA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aAB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aBA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aBB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aCA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aCB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHumanShow
DYRK1ADYRKCMGC6t6aDA-HumanShow
DYRK1ADYRKCMGC6t6aDB-HumanShow
DYRK1ADYRKCMGC6uipA4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHumanShow
DYRK1ADYRKCMGC6uipB4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHumanShow
DYRK1ADYRKCMGC6uipC4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHumanShow
DYRK1ADYRKCMGC6uwyAA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyAB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyBA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyBB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyCA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyCB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyDA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6uwyDB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHumanShow
DYRK1ADYRKCMGC6yf8A~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHumanShow
DYRK1ADYRKCMGC6yf8B~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHumanShow
DYRK1ADYRKCMGC6yf8C~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHumanShow
DYRK1ADYRKCMGC6yf8D~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHumanShow
DYRK1ADYRKCMGC7a4oAphosphoaminophosphonic acid-adenylate esterHumanShow
DYRK1ADYRKCMGC7a4rAA2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHumanShow
DYRK1ADYRKCMGC7a4rAB2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHumanShow
DYRK1ADYRKCMGC7a4sA7-chlorothieno[3,2-c]pyridin-4-amineHumanShow
DYRK1ADYRKCMGC7a4wA6-(4-methoxyphenyl)pyrimidine-2,4-diamineHumanShow
DYRK1ADYRKCMGC7a4zA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHumanShow
DYRK1ADYRKCMGC7a51A4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHumanShow
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