PDB-code
Browse kinase entries (page 96 of 282)
First 92 93 94 PreviousLast100 99 98 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | DYRK1A | DYRK | CMGC | 6s11 | B | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s11 | B | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s14 | A | A | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s14 | A | B | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s17 | A | A | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s17 | A | B | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1b | A | A | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1b | A | B | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1h | A | A | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1h | A | B | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | A | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | A | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | B | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | B | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | C | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | C | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | D | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1i | D | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1j | A | A | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6s1j | A | B | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | A | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | A | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | B | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | B | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | C | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | C | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | D | A | - | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6t6a | D | B | - | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uip | A | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6uip | B | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6uip | C | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6uwy | A | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | A | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | B | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | B | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | C | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | C | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | D | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6uwy | D | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 6yf8 | A | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6yf8 | B | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6yf8 | C | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 6yf8 | D | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a4o | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a4r | A | A | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a4r | A | B | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a4s | A | 7-chlorothieno[3,2-c]pyridin-4-amine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a4w | A | 6-(4-methoxyphenyl)pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a4z | A | 3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a51 | A | 4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | ![]() |


