PDB-code
Search results (14 entries covering 7 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhg | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() | |
![]() | PRKAA1 (AMPKa1) | CAMKL | CAMK | 7m74 | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() | |
![]() | ACVR1 (ALK2) | STKR | TKL | 3h9r | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() | |
![]() | ACVR1 (ALK2) | STKR | TKL | 4c02 | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | ACVR1 (ALK2) | STKR | TKL | 4c02 | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 6gvx | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 6gvx | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 6gvx | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | MELK | CAMKL | CAMK | 6gvx | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |
![]() | PRKAA2 (AMPKa2) | CAMKL | CAMK | 3aqv | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() | |
![]() | ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | Show | ![]() |


