Search results (14 entries covering 7 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PRKAA1 (AMPKa1)CAMKLCAMK7jhgA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
PRKAA1 (AMPKa1)CAMKLCAMK7m74A6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR1 (ALK2)STKRTKL3h9rA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR1 (ALK2)STKRTKL4c02AB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR1 (ALK2)STKRTKL4c02AA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR2A (ACTR2)STKRTKL3q4tBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR2A (ACTR2)STKRTKL3q4tAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR2A (ACTR2)STKRTKL3q4tAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
MELKCAMKLCAMK6gvxBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
MELKCAMKLCAMK6gvxAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
MELKCAMKLCAMK6gvxBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
MELKCAMKLCAMK6gvxAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
PRKAA2 (AMPKa2)CAMKLCAMK3aqvA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow
ACVR2A (ACTR2)STKRTKL3q4tBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHumanShow