Search results (5 entries covering 5 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
SIK3 (QSK)CAMKLCAMK8r4qA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHumanShow
SIK3 (QSK)CAMKLCAMK8r4uA8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHumanShow
SIK3 (QSK)CAMKLCAMK8r4vA1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]ureaHumanShow
SIK3 (QSK)CAMKLCAMK8r4oA2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamideHumanShow
SIK3 (QSK)CAMKLCAMK8okuA~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamideHumanShow