Search results (19 entries covering 8 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DCLK1DCAMKLCAMK6kyrBB-HumanShow
DCLK1DCAMKLCAMK6kyqAA-HumanShow
DCLK1DCAMKLCAMK5jzjBAamp phosphoramidateHumanShow
DCLK1DCAMKLCAMK5jznA5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHumanShow
DCLK1DCAMKLCAMK5jzjABamp phosphoramidateHumanShow
DCLK1DCAMKLCAMK5jznB5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHumanShow
DCLK1DCAMKLCAMK7f3gA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHumanShow
DCLK1DCAMKLCAMK6kyrAA-HumanShow
DCLK1DCAMKLCAMK6kyrBA-HumanShow
DCLK1DCAMKLCAMK7kxwA2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
DCLK1DCAMKLCAMK6kyqAB-HumanShow
DCLK1DCAMKLCAMK5jzjBBamp phosphoramidateHumanShow
DCLK1DCAMKLCAMK6kyrAB-HumanShow
DCLK1DCAMKLCAMK6kyqBB-HumanShow
DCLK1DCAMKLCAMK7kx6A2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
DCLK1DCAMKLCAMK6kyqBA-HumanShow
DCLK1DCAMKLCAMK5jzjAAamp phosphoramidateHumanShow
DCLK1DCAMKLCAMK7kxwB2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
DCLK1DCAMKLCAMK7kx8A5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow