PDB-code
Search results (40 entries covering 24 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | DYRK2 | DYRK | CMGC | 5lxd | B | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show |  |
| DYRK2 | DYRK | CMGC | 7dh3 | A | 2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 5ztn | B | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7ejv | B | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | Show | |
| DYRK2 | DYRK | CMGC | 7ejv | B | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dhk | A | 2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 6hdr | A | A | curcumin | Human | Show | |
| DYRK2 | DYRK | CMGC | 5lxc | B | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 3kvw | A | B | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | Show | |
| DYRK2 | DYRK | CMGC | 7akh | A | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 6hdp | A | B | scorzodihydrostilbene a | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dh9 | A | [2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanol | Human | Show | | |
| DYRK2 | DYRK | CMGC | 4azf | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | |
| DYRK2 | DYRK | CMGC | 5ztn | A | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7dhn | A | 7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinoline | Human | Show | | |
| DYRK2 | DYRK | CMGC | 5lxd | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 3k2l | A | B | - | Human | Show | |
| DYRK2 | DYRK | CMGC | 3k2l | A | A | - | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dho | A | 2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7ejv | A | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dl6 | A | [2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7ejv | A | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | Show | |
| DYRK2 | DYRK | CMGC | 4azf | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dg4 | A | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 6hdr | A | B | curcumin | Human | Show | |
| DYRK2 | DYRK | CMGC | 5lxd | B | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 7akf | A | B | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | |
| DYRK2 | DYRK | CMGC | 5lxc | A | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dhc | A | 4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7djo | A | [2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | Show | | |
| DYRK2 | DYRK | CMGC | 5lxd | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 7akf | A | A | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | |
| DYRK2 | DYRK | CMGC | 5lxc | A | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 6k0j | A | 3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amine | Human | Show | | |
| DYRK2 | DYRK | CMGC | 8hlt | A | (6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanone | Human | Show | | |
| DYRK2 | DYRK | CMGC | 5lxc | B | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | Show | |
| DYRK2 | DYRK | CMGC | 6hdp | A | A | scorzodihydrostilbene a | Human | Show | |
| DYRK2 | DYRK | CMGC | 7dhv | A | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acid | Human | Show | | |
| DYRK2 | DYRK | CMGC | 7dhh | A | [9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanol | Human | Show | | |
| DYRK2 | DYRK | CMGC | 3kvw | A | A | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | Show | |
