Search results (29 entries covering 9 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PRPF4B (PRP4)DYRKCMGC4ijpBA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpBB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4iirAAphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4ianA-HumanShow
PRPF4B (PRP4)DYRKCMGC4iirABphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjAA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjAB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcAAadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjBA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4iirBBphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcBBadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjCB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ianB-HumanShow
PRPF4B (PRP4)DYRKCMGC8h6eH-HumanShow
PRPF4B (PRP4)DYRKCMGC8h6jHB-HumanShow
PRPF4B (PRP4)DYRKCMGC8h6jHA-HumanShow
PRPF4B (PRP4)DYRKCMGC6pjjCA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pk6AB4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpAA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjDA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC4iirBAphosphoaminophosphonic acid-adenylate esterHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcBAadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4ifcABadenosine-5'-diphosphateHumanShow
PRPF4B (PRP4)DYRKCMGC4ijpAB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6cnhAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjDB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6cnhAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pjjBB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow
PRPF4B (PRP4)DYRKCMGC6pk6AA4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHumanShow