PDB-code
Search results (18 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6ylc | C | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yll | B | - | Human | Show | ![]() | |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6ylc | A | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6yll | A | ~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamine | Human | Show | ![]() | |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | A | - | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | B | - | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | A | - | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6ylc | D | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | ![]() | |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | B | - | Human | Show | ![]() |
![]() | MAPK6 (Erk3) | MAPK | CMGC | 6ylc | B | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | Show | ![]() |


