Search results (18 entries covering 4 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAPK6 (Erk3)MAPKCMGC6ykyDA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ylcC5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyCB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6yllB-HumanShow
MAPK6 (Erk3)MAPKCMGC6ykyBB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyCA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyAA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyDB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyAB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6ylcA5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHumanShow
MAPK6 (Erk3)MAPKCMGC6ykyBA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHumanShow
MAPK6 (Erk3)MAPKCMGC6yllA~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamineHumanShow
MAPK6 (Erk3)MAPKCMGC7aqbBA-HumanShow
MAPK6 (Erk3)MAPKCMGC7aqbAB-HumanShow
MAPK6 (Erk3)MAPKCMGC7aqbAA-HumanShow
MAPK6 (Erk3)MAPKCMGC6ylcD5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHumanShow
MAPK6 (Erk3)MAPKCMGC7aqbBB-HumanShow
MAPK6 (Erk3)MAPKCMGC6ylcB5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHumanShow