Search results (10 entries covering 6 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
EIF2AK4 (GCN2)PEKOther6n3lAAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHumanShow
EIF2AK4 (GCN2)PEKOther8t7tAA-HumanShow
EIF2AK4 (GCN2)PEKOther6n3nAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamideHumanShow
EIF2AK4 (GCN2)PEKOther7qwkA(2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamideHumanShow
EIF2AK4 (GCN2)PEKOther6n3lBAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHumanShow
EIF2AK4 (GCN2)PEKOther6n3lBBn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHumanShow
EIF2AK4 (GCN2)PEKOther7qq6A4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
EIF2AK4 (GCN2)PEKOther8t7tAB-HumanShow
EIF2AK4 (GCN2)PEKOther6n3oAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamideHumanShow
EIF2AK4 (GCN2)PEKOther6n3lABn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHumanShow