PDB-code
Search results (22 entries covering 13 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | EIF2AK3 (PEK) | PEK | Other | 4g31 | A | B | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone | Human | Show |  |
| EIF2AK3 (PEK) | PEK | Other | 4x7l | A | B | 4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7j | A | A | 2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 8eq9 | A | B | (2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7h | A | B | n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4g34 | A | B | 1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanone | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7k | A | B | 4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7o | A | B | 1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 8eqe | A | (2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetamide | Human | Show | | |
| EIF2AK3 (PEK) | PEK | Other | 4x7n | A | B | 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7j | A | B | 2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7k | A | A | 4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7n | A | A | 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4g31 | A | A | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7o | A | A | 1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 7mf0 | A | 2-amino-n-cyclopropyl-5-(4-{[(2r)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamide | Human | Show | | |
| EIF2AK3 (PEK) | PEK | Other | 8eqd | A | (2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | Show | | |
| EIF2AK3 (PEK) | PEK | Other | 8eq9 | A | A | (2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4x7h | A | A | n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4m7i | A | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-1h-indol-1-yl]-2-(6-methylpyridin-2-yl)ethanone | Human | Show | | |
| EIF2AK3 (PEK) | PEK | Other | 4x7l | A | A | 4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | Show | |
| EIF2AK3 (PEK) | PEK | Other | 4g34 | A | A | 1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanone | Human | Show | |
