PDB-code
Search results (13 entries covering 8 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | TEK (TIE2) | Tie | TK | 2oo8 | X | n-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamide | Human | Show |  | |
| TEK (TIE2) | Tie | TK | 2wqb | A | 2-[3-(cyclohexylmethyl)-5-phenyl-imidazol-4-yl]-[1,3]thiazolo[4,5-e]pyrimidin-7-amine | Human | Show | | |
| TEK (TIE2) | Tie | TK | 6mwe | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 1fvr | B | - | Human | Show | | |
| TEK (TIE2) | Tie | TK | 6mwe | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 4x3j | A | 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5h)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | Show | | |
| TEK (TIE2) | Tie | TK | 3l8p | A | 2-methyl-11-(1-methylethyl)-8-[(2s)-tetrahydro-2h-pyran-2-yl]-2,11,12,13-tetrahydro-4h-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2p4i | A | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 6mwe | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
| TEK (TIE2) | Tie | TK | 2p4i | B | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 1fvr | A | - | Human | Show | | |
| TEK (TIE2) | Tie | TK | 2osc | A | n-{4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]phenyl}-3-(trifluoromethyl)benzamide | Human | Show | | |
| TEK (TIE2) | Tie | TK | 6mwe | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | Show | |
