Search results (26 entries covering 20 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
RPS6KB1 (p70S6K)RSKAGC7n91A4-{[(1s)-1-(3-fluorophenyl)-2-(methylamino)ethyl]amino}quinazoline-8-carboxamideHumanShow
RPS6KB1 (p70S6K)RSKAGC7n93AA4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamideHumanShow
RPS6KB1 (p70S6K)RSKAGC4l46A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC4l3lA2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC4l43A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC3we4A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf7AB1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamideHumanShow
RPS6KB1 (p70S6K)RSKAGC4l42A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC4l3jA2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC7n93AB4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamideHumanShow
RPS6KB1 (p70S6K)RSKAGC3a61AstaurosporineHumanShow
RPS6KB1 (p70S6K)RSKAGC4l45A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf5AB4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidineHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf6AB4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidineHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf7AA1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamideHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf8A2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl 7,8,9,10-tetrahydro-6h-cyclohepta[b]quinoline-11-carboxylateHumanShow
RPS6KB1 (p70S6K)RSKAGC3a62AstaurosporineHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf5AA4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidineHumanShow
RPS6KB1 (p70S6K)RSKAGC4rlpA[(amino-kappan)methanethiolato](3-fluoro-9-methoxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(n-methyl-1,4,7-trithiecan-9-amine-kappa~3~s~1~,s~4~,s~7~)rutheniumHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf9A(2s)-1-oxo-1-[(4-sulfamoylphenyl)amino]propan-2-yl (2s)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylateHumanShow
RPS6KB1 (p70S6K)RSKAGC4rloA[(amino-kappan)methanethiolato](3-fluoro-9-hydroxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)rutheniumHumanShow
RPS6KB1 (p70S6K)RSKAGC3a60BstaurosporineHumanShow
RPS6KB1 (p70S6K)RSKAGC3a60AstaurosporineHumanShow
RPS6KB1 (p70S6K)RSKAGC3wf6AA4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidineHumanShow
RPS6KB1 (p70S6K)RSKAGC4l44A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHumanShow
RPS6KB1 (p70S6K)RSKAGC4rloBstaurosporineHumanShow