PDB-code
Search results (38 entries covering 11 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 7szr | A | A | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 7szr | A | B | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | B | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | A | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | B | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | A | - | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | B | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | A | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | A | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | B | - | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | B | - | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | B | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | A | - | Mouse | Show | ![]() |
![]() | Map3k14 (NIK) | STE-Unique | STE | 6myn | A | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | Show | ![]() |


