PDB-code
Browse kinase entries (page 101 of 282)
First 97 98 99 PreviousLast105 104 103 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | EGFR | EGFR | TK | 4lqm | A | n-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4lrm | A | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4lrm | B | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4lrm | C | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4lrm | D | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4lrm | E | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4r3p | A | - | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4r3r | A | - | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4r5s | A | n-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4riw | B | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4riw | D | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rix | B | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rix | D | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4riy | B | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4riy | D | adenosine-5'-diphosphate | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rj4 | A | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1-(propan-2-yl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rj5 | A | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rj6 | A | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-3h-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4rj7 | A | A | 2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4rj7 | A | B | 2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamide | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4rj8 | A | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4tks | A | - | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4wd5 | A | n-{2-methyl-5-[2-oxo-9-(1h-pyrazol-4-yl)benzo[h][1,6]naphthyridin-1(2h)-yl]phenyl}propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4wd5 | B | - | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4wkq | A | A | gefitinib | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4wkq | A | B | gefitinib | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4wrg | A | A | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4wrg | A | B | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zau | A | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 4zjv | A | A | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zjv | A | B | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zjv | B | A | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zjv | B | B | - | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | B | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | B | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | C | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | C | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | D | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 4zse | D | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 5c8k | A | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5c8m | A | 2-methyl-n-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5c8n | A | n-{2-[4-(2-aminoethyl)-4-methoxypiperidin-1-yl]pyrimidin-4-yl}-2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5cal | A | 2,2-dimethyl-3-[(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)amino]propanamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5can | A | (3r)-3-methyl-1-(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)pyrrolidine-3-carboxamide | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5cao | A | n~2~-[2-methyl-2-(methylsulfonyl)propyl]-n~4~-[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]pyrimidine-2,4-diamine | Human | Show | ![]() | |
![]() | EGFR | EGFR | TK | 5cap | A | A | 2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 5cap | A | B | 2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() |
![]() | EGFR | EGFR | TK | 5caq | A | n-[2-[(3r,4s)-3-fluoranyl-4-methoxy-piperidin-1-yl]pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | Show | ![]() |


