Browse kinase entries (page 101 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
EGFREGFRTK4lqmAn-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamideHumanShow
EGFREGFRTK4lrmAn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHumanShow
EGFREGFRTK4lrmBn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHumanShow
EGFREGFRTK4lrmCn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHumanShow
EGFREGFRTK4lrmDn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHumanShow
EGFREGFRTK4lrmEn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHumanShow
EGFREGFRTK4r3pA-HumanShow
EGFREGFRTK4r3rA-HumanShow
EGFREGFRTK4r5sAn-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamideHumanShow
EGFREGFRTK4riwBadenosine-5'-diphosphateHumanShow
EGFREGFRTK4riwDadenosine-5'-diphosphateHumanShow
EGFREGFRTK4rixBadenosine-5'-diphosphateHumanShow
EGFREGFRTK4rixDadenosine-5'-diphosphateHumanShow
EGFREGFRTK4riyBadenosine-5'-diphosphateHumanShow
EGFREGFRTK4riyDadenosine-5'-diphosphateHumanShow
EGFREGFRTK4rj4An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1-(propan-2-yl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHumanShow
EGFREGFRTK4rj5An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHumanShow
EGFREGFRTK4rj6An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-3h-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK4rj7AA2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamideHumanShow
EGFREGFRTK4rj7AB2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamideHumanShow
EGFREGFRTK4rj8A1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHumanShow
EGFREGFRTK4tksA-HumanShow
EGFREGFRTK4wd5An-{2-methyl-5-[2-oxo-9-(1h-pyrazol-4-yl)benzo[h][1,6]naphthyridin-1(2h)-yl]phenyl}propanamideHumanShow
EGFREGFRTK4wd5B-HumanShow
EGFREGFRTK4wkqAAgefitinibHumanShow
EGFREGFRTK4wkqABgefitinibHumanShow
EGFREGFRTK4wrgAA-HumanShow
EGFREGFRTK4wrgAB-HumanShow
EGFREGFRTK4zauAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHumanShow
EGFREGFRTK4zjvAA-HumanShow
EGFREGFRTK4zjvAB-HumanShow
EGFREGFRTK4zjvBA-HumanShow
EGFREGFRTK4zjvBB-HumanShow
EGFREGFRTK4zseAAphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseABphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseBAphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseBBphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseCAphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseCBphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseDAphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK4zseDBphosphoaminophosphonic acid-adenylate esterHumanShow
EGFREGFRTK5c8kA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK5c8mA2-methyl-n-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK5c8nAn-{2-[4-(2-aminoethyl)-4-methoxypiperidin-1-yl]pyrimidin-4-yl}-2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK5calA2,2-dimethyl-3-[(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)amino]propanamideHumanShow
EGFREGFRTK5canA(3r)-3-methyl-1-(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)pyrrolidine-3-carboxamideHumanShow
EGFREGFRTK5caoAn~2~-[2-methyl-2-(methylsulfonyl)propyl]-n~4~-[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]pyrimidine-2,4-diamineHumanShow
EGFREGFRTK5capAA2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK5capAB2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHumanShow
EGFREGFRTK5caqAn-[2-[(3r,4s)-3-fluoranyl-4-methoxy-piperidin-1-yl]pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHumanShow
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