Browse kinase entries (page 119 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
ERN1 (IRE1)IREOther6w3bA-HumanShow
ERN1 (IRE1)IREOther6w3cA-HumanShow
ERN1 (IRE1)IREOther6w3cB-HumanShow
ERN1 (IRE1)IREOther6w3cC-HumanShow
ERN1 (IRE1)IREOther6w3cD-HumanShow
ERN1 (IRE1)IREOther6w3eAmethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHumanShow
ERN1 (IRE1)IREOther6w3eBmethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHumanShow
ERN1 (IRE1)IREOther6w3kA4-[5-[2,6-bis(fluoranyl)phenyl]-2~{h}-pyrazolo[3,4-b]pyridin-3-yl]-2-(4-oxidanylpiperidin-1-yl)-1~{h}-pyrimidin-6-oneHumanShow
ERN1 (IRE1)IREOther6xdbA4-amino-n-(6-chloro-2-fluoro-3-{[(2-fluorophenyl)sulfonyl]amino}phenyl)-6-(1,3-dimethyl-1h-pyrazol-4-yl)quinazoline-8-carboxamideHumanShow
ERN1 (IRE1)IREOther6xddA4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamideHumanShow
ERN1 (IRE1)IREOther6xddB4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamideHumanShow
ERN1 (IRE1)IREOther6xdfBA-HumanShow
ERN1 (IRE1)IREOther6xdfBB-HumanShow
ERN1 (IRE1)IREOther7bmkAA2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamideHumanShow
ERN1 (IRE1)IREOther7bmkAB2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamideHumanShow
FESFerTK3bkbAAstaurosporineHumanShow
FESFerTK3bkbABstaurosporineHumanShow
FESFerTK3bkbACstaurosporineHumanShow
FESFerTK3cblAAstaurosporineHumanShow
FESFerTK3cblABstaurosporineHumanShow
FESFerTK3cd3AAstaurosporineHumanShow
FESFerTK3cd3ABstaurosporineHumanShow
FESFerTK4e93AA5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHumanShow
FESFerTK4e93AB5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHumanShow
FESFerTK6jmfA6-{[(1r,2s)-2-aminocyclohexyl]amino}-5-cyano-2-[(3-methylphenyl)amino]pyridine-3-carboxamideHumanShow
FGFR1FGFRTK1agwAA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK1agwAB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK1agwBA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK1agwBB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK1fgiAA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK1fgiAB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK1fgiBA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK1fgiBB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK1fgkAA-HumanShow
FGFR1FGFRTK1fgkAB-HumanShow
FGFR1FGFRTK1fgkBA-HumanShow
FGFR1FGFRTK1fgkBB-HumanShow
FGFR1FGFRTK2fgiA1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHumanShow
FGFR1FGFRTK2fgiB1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHumanShow
FGFR1FGFRTK3c4fAA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK3c4fAB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK3c4fBA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK3c4fBB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK3gqiAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR1FGFRTK3gqlA(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK3gqlB(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK3gqlC(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK3js2A5-(2-thienyl)nicotinic acidHumanShow
FGFR1FGFRTK3js2B5-(2-thienyl)nicotinic acidHumanShow
FGFR1FGFRTK3kxxA-HumanShow
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