PDB-code
Browse kinase entries (page 119 of 282)
First 115 116 117 PreviousLast123 122 121 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | ERN1 (IRE1) | IRE | Other | 6w3b | A | - | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3c | A | - | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3c | B | - | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3c | C | - | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3c | D | - | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3e | A | methyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3e | B | methyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6w3k | A | 4-[5-[2,6-bis(fluoranyl)phenyl]-2~{h}-pyrazolo[3,4-b]pyridin-3-yl]-2-(4-oxidanylpiperidin-1-yl)-1~{h}-pyrimidin-6-one | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6xdb | A | 4-amino-n-(6-chloro-2-fluoro-3-{[(2-fluorophenyl)sulfonyl]amino}phenyl)-6-(1,3-dimethyl-1h-pyrazol-4-yl)quinazoline-8-carboxamide | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6xdd | A | 4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamide | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6xdd | B | 4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamide | Human | Show | ![]() | |
![]() | ERN1 (IRE1) | IRE | Other | 6xdf | B | A | - | Human | Show | ![]() |
![]() | ERN1 (IRE1) | IRE | Other | 6xdf | B | B | - | Human | Show | ![]() |
![]() | ERN1 (IRE1) | IRE | Other | 7bmk | A | A | 2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamide | Human | Show | ![]() |
![]() | ERN1 (IRE1) | IRE | Other | 7bmk | A | B | 2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamide | Human | Show | ![]() |
![]() | FES | Fer | TK | 3bkb | A | A | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3bkb | A | B | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3bkb | A | C | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3cbl | A | A | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3cbl | A | B | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3cd3 | A | A | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 3cd3 | A | B | staurosporine | Human | Show | ![]() |
![]() | FES | Fer | TK | 4e93 | A | A | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FES | Fer | TK | 4e93 | A | B | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | Show | ![]() |
![]() | FES | Fer | TK | 6jmf | A | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-5-cyano-2-[(3-methylphenyl)amino]pyridine-3-carboxamide | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 1agw | A | A | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1agw | A | B | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1agw | B | A | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1agw | B | B | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgi | A | A | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgi | A | B | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgi | B | A | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgi | B | B | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgk | A | A | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgk | A | B | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgk | B | A | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 1fgk | B | B | - | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 2fgi | A | 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 2fgi | B | 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3c4f | A | A | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3c4f | A | B | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3c4f | B | A | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3c4f | B | B | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | FGFR1 | FGFR | TK | 3gqi | A | phosphomethylphosphonic acid adenylate ester | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3gql | A | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3gql | B | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3gql | C | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3js2 | A | 5-(2-thienyl)nicotinic acid | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3js2 | B | 5-(2-thienyl)nicotinic acid | Human | Show | ![]() | |
![]() | FGFR1 | FGFR | TK | 3kxx | A | - | Human | Show | ![]() |


